Quinoline derivative MC1626, a putative GCN5 histone acetyltransferase (HAT) inhibitor, exhibits HAT-independent activity against Toxoplasma gondii.
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Toxoplasma histone acetylation remodelers as novel drug targetsProtein lysine acetylation by p300/CBPGarcinol Inhibits GCN5-Mediated Lysine Acetyltransferase Activity and Prevents Replication of the Parasite Toxoplasma gondii.Review of Experimental Compounds Demonstrating Anti-Toxoplasma Activity.Histone acetyltransferase inhibitors and preclinical studies.A Systematic Review of In vitro and In vivo Activities of Anti-Toxoplasma Drugs and Compounds (2006-2016).Screening for small molecule inhibitors of Toxoplasma gondii.
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Q22305931-CA8B7E81-5461-48C0-BD9C-4717B085D10BQ27021749-12416425-EE0D-491B-B75D-5850C8B770B8Q36729982-B795DEA8-6762-4C8B-B228-2C3DDC3B72D6Q37428599-3D14A9CA-4647-4B89-B015-BBDBF9627043Q37497374-67189C4D-8317-4D83-A027-00284AB881AEQ37594988-5DE93E34-06EB-4E49-A8C8-EACDEA48DF4DQ38045464-CD518B98-3C0F-4694-8922-2BA646BD57E4
P2860
Quinoline derivative MC1626, a putative GCN5 histone acetyltransferase (HAT) inhibitor, exhibits HAT-independent activity against Toxoplasma gondii.
description
2006 nî lūn-bûn
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2006年の論文
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name
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@ast
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@en
type
label
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@ast
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@en
prefLabel
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@ast
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@en
P2093
P2860
P356
P1476
Quinoline derivative MC1626, a ...... ity against Toxoplasma gondii.
@en
P2093
Aaron T Smith
Meredith R Livingston
Sherry F Queener
William J Sullivan
P2860
P304
P356
10.1128/AAC.01256-06
P407
P577
2006-12-18T00:00:00Z