Relative affinities of drugs acting at cholinoceptors in displacing agonist and antagonist radioligands: the NMS/Oxo-M ratio as an index of efficacy at cortical muscarinic receptors.
about
Rotigotine is a potent agonist at dopamine D1 receptors as well as at dopamine D2 and D3 receptorsDifferential modulation by GTPgammaS of agonist and inverse agonist binding to h5-HT(1A) receptors revealed by [3H]-WAY100,635Functional effects of the muscarinic receptor agonist, xanomeline, at 5-HT1 and 5-HT2 receptorsMuscarinic receptor/G-protein coupling is reduced in the dorsomedial striatum of cognitively impaired aged rats.Relationship between inhibition of cyclic AMP production in Chinese hamster ovary cells expressing the rat D2(444) receptor and antagonist/agonist binding ratios.A novel series of non-quaternary oxadiazoles acting as full agonists at muscarinic receptors.Mixed nicotinic and muscarinic features of cholinergic receptor coupled to secretion in bovine chromaffin cellsAntinociceptive and toxic effects of (+)-epibatidine oxalate attributable to nicotinic agonist activity.L-689,660, a novel cholinomimetic with functional selectivity for M1 and M3 muscarinic receptors.Inverse agonist activity of pirenzepine at M2 muscarinic acetylcholine receptors.Nad-299 antagonises 5-HT-stimulated and spiperone-inhibited [35S]GTPgammaS binding in cloned 5-HT1A receptors.The cholinergic pharmacology of tetrahydroaminoacridine in vivo and in vitro.5-HT(1A) receptor agonist-antagonist binding affinity difference as a measure of intrinsic activity in recombinant and native tissue systems.Preconditioning stimuli that augment chromaffin cell secretion.Circadian rhythm in muscarinic receptor subtypes in rat forebrain.Evaluation of an agonist index: affinity ratio for compounds active on muscarinic cholinergic M2 receptors.SR 46559A: a novel and potent muscarinic compound with no cholinergic syndrome.Effects of serotonergic denervation on the density and plasticity of brain muscarinic receptors in the rat.Loss of high-affinity agonist binding to M1 muscarinic receptors in Alzheimer's disease: implications for the failure of cholinergic replacement therapies.Analogues of carbacholine: synthesis and relationship between structure and affinity for muscarinic and nicotinic acetylcholine receptors.
P2860
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P2860
Relative affinities of drugs acting at cholinoceptors in displacing agonist and antagonist radioligands: the NMS/Oxo-M ratio as an index of efficacy at cortical muscarinic receptors.
description
1988 nî lūn-bûn
@nan
1988年の論文
@ja
1988年論文
@yue
1988年論文
@zh-hant
1988年論文
@zh-hk
1988年論文
@zh-mo
1988年論文
@zh-tw
1988年论文
@wuu
1988年论文
@zh
1988年论文
@zh-cn
name
Relative affinities of drugs a ...... cortical muscarinic receptors.
@ast
Relative affinities of drugs a ...... cortical muscarinic receptors.
@en
type
label
Relative affinities of drugs a ...... cortical muscarinic receptors.
@ast
Relative affinities of drugs a ...... cortical muscarinic receptors.
@en
prefLabel
Relative affinities of drugs a ...... cortical muscarinic receptors.
@ast
Relative affinities of drugs a ...... cortical muscarinic receptors.
@en
P2860
P1476
Relative affinities of drugs a ...... cortical muscarinic receptors.
@en
P2093
Freedman SB
P2860
P304
P356
10.1111/J.1476-5381.1988.TB11451.X
P407
P577
1988-02-01T00:00:00Z