Synthesis and pharmacological characterization of a novel sigma receptor ligand with improved metabolic stability and antagonistic effects against methamphetamine
about
SN79, a sigma receptor antagonist, attenuates methamphetamine-induced astrogliosis through a blockade of OSMR/gp130 signaling and STAT3 phosphorylationSigma-1 receptor chaperones in neurodegenerative and psychiatric disordersUltra-performance liquid chromatography tandem mass spectrometry method for the determination of AZ66, a sigma receptor ligand, in rat plasma and its application to in vivo pharmacokinetics.Sigma receptor antagonists attenuate acute methamphetamine-induced hyperthermia by a mechanism independent of IL-1β mRNA expression in the hypothalamus.Blockade of Cocaine or σ Receptor Agonist Self Administration by Subtype-Selective σ Receptor Antagonists.Novel Sigma-1 receptor antagonists: from opioids to small molecules: what is new?The sigma-1 receptor as a regulator of dopamine neurotransmission: A potential therapeutic target for methamphetamine addiction.
P2860
Q23918033-3D3763F3-1677-4665-8FAB-57D62AD3CA74Q33920251-EE1B6381-B6C0-48C8-A021-676B6E8EB5D0Q34005371-613A1B94-CFF2-403F-8F09-678879BEEFEDQ37052573-25307081-F728-4B63-BA22-F7407EF074E2Q37062588-57EB86EB-9663-4CF4-858E-7CAE23F2554AQ47353437-493F2C62-1E99-4A3B-AC9B-56D33B2852B6Q47845016-519DC7B1-8B5F-42EB-B923-9C26F000D6AD
P2860
Synthesis and pharmacological characterization of a novel sigma receptor ligand with improved metabolic stability and antagonistic effects against methamphetamine
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Synthesis and pharmacological ...... ffects against methamphetamine
@ast
Synthesis and pharmacological ...... ffects against methamphetamine
@en
type
label
Synthesis and pharmacological ...... ffects against methamphetamine
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Synthesis and pharmacological ...... ffects against methamphetamine
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prefLabel
Synthesis and pharmacological ...... ffects against methamphetamine
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Synthesis and pharmacological ...... ffects against methamphetamine
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P2093
P2860
P1433
P1476
Synthesis and pharmacological ...... ffects against methamphetamine
@en
P2093
Ahmed H Abdelazeem
Bonnie A Avery
Christophe Mesangeau
Christopher R McCurdy
Matthew J Robson
Michael J Seminerio
Rae R Matsumoto
Seshulatha Jamalapuram
P2860
P2888
P356
10.1208/S12248-011-9311-8
P407
P577
2011-12-20T00:00:00Z
P5875
P6179
1045722268