Ligand-specific roles for transmembrane 5 serine residues in the binding and efficacy of dopamine D(1) receptor catechol agonists
about
Dopamine D1 receptor signaling: does GαQ-phospholipase C actually play a role?Structure and dynamics of DRD4 bound to an agonist and an antagonist using in silico approaches.SKF-83959 is not a highly-biased functionally selective D1 dopamine receptor ligand with activity at phospholipase CComputational analysis of C-reactive protein for assessment of molecular dynamics and interaction properties.Structural signatures of DRD4 mutants revealed using molecular dynamics simulations: Implications for drug targeting.Detailed analysis of biased histamine H₄ receptor signalling by JNJ 7777120 analogues.Impaired β-arrestin recruitment and reduced desensitization by non-catechol agonists of the D1 dopamine receptor.Functional roles of T3.37 and S5.46 in the activation mechanism of the dopamine D1 receptor.
P2860
Q26864383-038CB411-8185-4F6E-A65B-33F101107166Q30009287-D86374E9-3E53-4178-888D-06AD20286199Q30400003-88E0EB90-CC94-498F-9783-E04A1E4EA0F1Q37417484-337F7F53-302A-4A73-82B2-B2EB63E6F675Q38384318-33B40ED8-14F9-4DC8-96D0-F87C572F4D2FQ39204577-5CC6E1AA-EAF1-4159-946E-05E8BDAA9944Q49234399-DD0316C6-F506-4AFE-82B7-DA5FB8707078Q52694045-A02B3B3C-8490-49B1-876A-088F44502FE0
P2860
Ligand-specific roles for transmembrane 5 serine residues in the binding and efficacy of dopamine D(1) receptor catechol agonists
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年学术文章
@wuu
2012年学术文章
@zh-cn
2012年学术文章
@zh-hans
2012年学术文章
@zh-my
2012年学术文章
@zh-sg
2012年學術文章
@yue
2012年學術文章
@zh
2012年學術文章
@zh-hant
name
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@ast
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@en
type
label
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@ast
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@en
prefLabel
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@ast
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@en
P2093
P2860
P356
P1476
Ligand-specific roles for tran ...... (1) receptor catechol agonists
@en
P2093
Benjamin R Chemel
David E Nichols
Lisa A Bonner
Val J Watts
P2860
P304
P356
10.1124/MOL.111.077339
P577
2012-02-14T00:00:00Z