Molecular basis for binding and subtype selectivity of 1,4-benzodiazepine antagonist ligands of the cholecystokinin receptor.

Molecular basis for binding and subtype selectivity of 1,4-benzodiazepine antagonist ligands of the cholecystokinin receptor.

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http://www.wikidata.org/entity/Q36002904
Cholecystokinin-induced satiety, a key gut servomechanism that is affected by the membrane microenvironment of this receptorA type 1 cholecystokinin receptor mutant that mimics the dysfunction observed for wild type receptor in a high cholesterol environment.Development of a highly selective allosteric antagonist radioligand for the type 1 cholecystokinin receptor and elucidation of its molecular basis of bindingElimination of a cholecystokinin receptor agonist 'trigger' in an effort to develop positive allosteric modulators without intrinsic agonist activity.Impact of ursodeoxycholic acid on a CCK1R cholesterol-binding site may contribute to its positive effects in digestive function.Sensitivity of cholecystokinin receptors to membrane cholesterol content.Molecular Mechanism of Action of Triazolobenzodiazepinone Agonists of the Type 1 Cholecystokinin Receptor. Possible Cooperativity across the Receptor Homodimeric Complex.Direct demonstration of unique mode of natural peptide binding to the type 2 cholecystokinin receptor using photoaffinity labeling.Molecular basis for benzodiazepine agonist action at the type 1 cholecystokinin receptor.Metabolic Actions of the Type 1 Cholecystokinin Receptor: Its Potential as a Therapeutic Target.Beneficial effects of β-sitosterol on type 1 cholecystokinin receptor dysfunction induced by elevated membrane cholesterol.Structural studies on radiopharmaceutical DOTA-minigastrin analogue (CP04) complexes and their interaction with CCK2 receptor.Gastrin receptor pharmacology.
P2860

Molecular basis for binding and subtype selectivity of 1,4-benzodiazepine antagonist ligands of the cholecystokinin receptor.

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http://www.wikidata.org/entity/Q36002904
description
2012 nî lūn-bûn
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2012年の論文
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2012年論文
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2012年論文
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2012年論文
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2012年論文
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2012年論文
@zh-tw
2012年论文
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2012年论文
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2012年论文
@zh-cn
name
Molecular basis for binding an ...... the cholecystokinin receptor.
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Molecular basis for binding an ...... the cholecystokinin receptor.
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Molecular basis for binding an ...... the cholecystokinin receptor.
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Molecular basis for binding an ...... the cholecystokinin receptor.
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Molecular basis for binding an ...... the cholecystokinin receptor.
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Molecular basis for binding an ...... the cholecystokinin receptor.
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P1476
P2093
P2860
P304
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Molecular basis for binding an ...... the cholecystokinin receptor.
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P698
P921
P932