Bicyclic core estrogens as full antagonists: synthesis, biological evaluation and structure-activity relationships of estrogen receptor ligands based on bridged oxabicyclic core arylsulfonamides.
about
Predictive features of ligand-specific signaling through the estrogen receptorThiophene-core estrogen receptor ligands having superagonist activity.Full antagonism of the estrogen receptor without a prototypical ligand side chain.Triaryl-substituted Schiff bases are high-affinity subtype-selective ligands for the estrogen receptor.Adamantyl Antiestrogens with Novel Side Chains Reveal a Spectrum of Activities in Suppressing Estrogen Receptor Mediated Activities in Breast Cancer Cells.Oxabicycloheptene Sulfonate Protects Against β-Amyloid-induced Toxicity by Activation of PI3K/Akt and ERK Signaling Pathways Via GPER1 in C6 Cells.Synthesis and antitumor evaluation of novel sulfonylcycloureas derived from nitrogen mustard.Selenophenes: Introducing a New Element into the Core of Non-Steroidal Estrogen Receptor Ligands.
P2860
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P2860
Bicyclic core estrogens as full antagonists: synthesis, biological evaluation and structure-activity relationships of estrogen receptor ligands based on bridged oxabicyclic core arylsulfonamides.
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年学术文章
@wuu
2012年学术文章
@zh-cn
2012年学术文章
@zh-hans
2012年学术文章
@zh-my
2012年学术文章
@zh-sg
2012年學術文章
@yue
2012年學術文章
@zh
2012年學術文章
@zh-hant
name
Bicyclic core estrogens as ful ...... icyclic core arylsulfonamides.
@ast
Bicyclic core estrogens as ful ...... icyclic core arylsulfonamides.
@en
type
label
Bicyclic core estrogens as ful ...... icyclic core arylsulfonamides.
@ast
Bicyclic core estrogens as ful ...... icyclic core arylsulfonamides.
@en
prefLabel
Bicyclic core estrogens as ful ...... icyclic core arylsulfonamides.
@ast
Bicyclic core estrogens as ful ...... icyclic core arylsulfonamides.
@en
P2093
P2860
P356
P1476
Bicyclic core estrogens as ful ...... bicyclic core arylsulfonamides
@en
P2093
Chen Zhang
Chune Dong
John A Katzenellenbogen
Kathryn E Carlson
Kendall W Nettles
Manghong Zhu
Sathish Srinivasan
Valerie Cavett
Yangfan Zheng
P2860
P304
P356
10.1039/C2OB26531A
P577
2012-11-01T00:00:00Z