Amphipathic benzenes are designed inhibitors of the estrogen receptor alpha/steroid receptor coactivator interaction
about
Sulindac-Derived RXRα Modulators Inhibit Cancer Cell Growth by Binding to a Novel SiteDevelopment of a novel molecular sensor for imaging estrogen receptor-coactivator protein-protein interactionsTetrahydro-iso-alpha Acids Antagonize Estrogen Receptor Alpha Activity in MCF-7 Breast Cancer CellsA set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator bindingBlocking estrogen signaling after the hormone: pyrimidine-core inhibitors of estrogen receptor-coactivator binding.LXXLL peptide converts transportan 10 to a potent inducer of apoptosis in breast cancer cells.Minireview: Not picking pockets: nuclear receptor alternate-site modulators (NRAMs)Identification of a New RXRα Antagonist Targeting the Coregulator-Binding Site.Alternative inhibition of androgen receptor signaling: peptidomimetic pyrimidines as direct androgen receptor/coactivator disruptors.Selectively targeting estrogen receptors for cancer treatment.A noncompetitive small molecule inhibitor of estrogen-regulated gene expression and breast cancer cell growth that enhances proteasome-dependent degradation of estrogen receptor {alpha}.Small molecule inhibitors as probes for estrogen and androgen receptor actionIn silico discovery and validation of potent small-molecule inhibitors targeting the activation function 2 site of human oestrogen receptor αA complex task? Direct modulation of transcription factors with small molecules.Synthesis of biphenyl proteomimetics as estrogen receptor-alpha coactivator binding inhibitors.Nonsteroidal bivalent estrogen ligands: an application of the bivalent concept to the estrogen receptor.Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor.Nuclear receptor coregulators as a new paradigm for therapeutic targeting.Beyond the ligand-binding pocket: targeting alternate sites in nuclear receptors.1,2,3-Triazole-based inhibitors of Porphyromonas gingivalis adherence to oral streptococci and biofilm formation.Estrogen receptor alpha/co-activator interaction assay: TR-FRETSynthesis of a tetrasubstituted tetrahydronaphthalene scaffold for α-helix mimicry via a MgBr2-catalyzed Friedel-Crafts epoxide cycloalkylation.Perfluoro-tert-butyl Homoserine Is a Helix-Promoting, Highly Fluorinated, NMR-Sensitive Aliphatic Amino Acid: Detection of the Estrogen Receptor·Coactivator Protein-Protein Interaction by 19F NMR.A Cell-Permeable Stapled Peptide Inhibitor of the Estrogen Receptor/Coactivator Interaction.Benzothiophenone Derivatives Targeting Mutant Forms of Estrogen Receptor-α in Hormone-Resistant Breast Cancers.Design, synthesis and conformational analyses of bifacial benzamide based foldamersStructure–activity relationship studies of miniproteins targeting the androgen receptor–coactivator interaction
P2860
Q27682952-02D91F01-FFFA-435B-8970-1B2C7B9B838AQ28482848-F957F17B-9B55-4B3D-8DEF-BB635D1ACAF9Q30383660-3D8E7DE5-32FB-4A57-9F92-996E7AB30EB1Q30857680-792BA41C-CF33-4C0E-B9FD-9FA418A827BEQ33368775-4BA320B0-E0AE-4851-B18E-DE2EB3E358DEQ33580471-B66E42DF-F633-4E6F-8FEA-4DE8B520DFBBQ33780204-B76CCB05-0195-48FA-ABF8-3B52349C64D7Q33889103-08F7951A-834D-4E13-B062-734346167F25Q34140002-573C1A0E-1E79-4DCD-853A-191E29FE1909Q34349374-A2A85370-19DD-491D-8859-AFA9EAE39201Q34438994-6BB1E697-BF6C-4AFE-9B24-B66587F91B59Q34575905-BFFB8E9F-4F52-4687-A536-E50A069C915FQ35180278-A24A9240-3773-4EFD-AE33-7F85F3541304Q35642431-68E38343-039D-4B94-B2A8-AD9CECD71666Q35687193-EBF85A8F-A004-4C16-9990-CFD8551B8A0CQ36781304-66B16E1F-7176-4C20-ADB8-D05BAB661513Q37036955-201ACB08-F88D-4230-B5BC-9E6A6E478B5DQ37217158-8B00D3AD-8AD4-45BD-B285-21EFEFBE518DQ38076345-B379B631-1E7F-4A9D-875A-BA9CC7D126D2Q40534514-87C891EE-12C6-4405-A894-E8F3E989C7BAQ41092895-7FD3BB76-D6C0-4C79-822A-9C80ED458F9AQ42062610-6B3CAEAB-7841-4705-AF99-763EB0EC7E0DQ48273411-AA633C50-F9AA-45D0-B204-56C9010B4A6DQ48295284-A7DFF879-DFB2-4262-8557-1CE54536E35FQ49805743-BADF8AF6-E5DE-4B18-9BAB-12B79C98CF18Q56830350-312BE860-9A1E-4E6B-8619-2525A9042774Q57531405-95345D01-FC26-4D99-8EA4-96228C7A802E
P2860
Amphipathic benzenes are designed inhibitors of the estrogen receptor alpha/steroid receptor coactivator interaction
description
2008 nî lūn-bûn
@nan
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
2008年论文
@zh
2008年论文
@zh-cn
name
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@ast
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@en
type
label
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@ast
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@en
prefLabel
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@ast
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@en
P2093
P2860
P356
P1433
P1476
Amphipathic benzenes are desig ...... ceptor coactivator interaction
@en
P2093
Jillian R Gunther
John A Katzenellenbogen
Margaret L Collins
Terry W Moore
P2860
P304
P356
10.1021/CB800056R
P577
2008-05-01T00:00:00Z