Intermolecular interactions identify ligand-selective activity of estrogen receptor alpha/beta dimers.
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Cyclopia extracts act as ERα antagonists and ERβ agonists, in vitro and in vivoIdentification of estrogen receptor dimer selective ligands reveals growth-inhibitory effects on cells that co-express ERα and ERβRegulation of estrogen receptor α N-terminus conformation and function by peptidyl prolyl isomerase Pin1Identification and characterization of a novel estrogenic ligand actinopolymorphol AGenome-wide dynamics of chromatin binding of estrogen receptors alpha and beta: mutual restriction and competitive site selection.Δ(9)-Tetrahydrocannabinol disrupts estrogen-signaling through up-regulation of estrogen receptor β (ERβ)Differential requirements of Hsp90 and DNA for the formation of estrogen receptor homodimers and heterodimers.Discovery and total synthesis of a new estrogen receptor heterodimerizing actinopolymorphol A from Actinopolymorpha rutilusEstrogen receptor beta selective nonsteroidal estrogens: seeking clinical indications.A dominant negative ERβ splice variant determines the effectiveness of early or late estrogen therapy after ovariectomy in ratsDevelopment of subtype-selective oestrogen receptor-based therapeutics.The role of hypothalamic estrogen receptors in metabolic regulation.Selectively targeting estrogen receptors for cancer treatment.Endocrine disrupting chemicals targeting estrogen receptor signaling: identification and mechanisms of action.Complex formation and interactions between transcription factors essential for human prolactin receptor gene transcription.Estrogen directly and specifically downregulates NaPi-IIa through the activation of both estrogen receptor isoforms (ERα and ERβ) in rat kidney proximal tubule.Evolutionary origins of the estrogen signaling system: insights from amphioxusAndrogens and estrogens in benign prostatic hyperplasia: past, present and future.Generation of stable reporter breast cancer cell lines for the identification of ER subtype selective ligands.Estrogen receptor-beta sensitizes breast cancer cells to the anti-estrogenic actions of endoxifenEstrogen-related Receptor β Reduces the Subnuclear Mobility of Estrogen Receptor α and Suppresses Estrogen-dependent Cellular Function.In vitro and in vivo molecular imaging of estrogen receptor α and β homo- and heterodimerization: exploration of new modes of receptor regulation.Divide and Conquer May Not Be the Optimal Approach to Retain the Desirable Estrogenic Attributes of the Cyclopia Nutraceutical Extract, SM6Met.17β-estradiol signaling and regulation of Sertoli cell functionReciprocal Regulation of ERα and ERβ Stability and Activity by Diptoindonesin G.Contribution of estrogen receptor subtypes, ERα, ERβ, and GPER1 in rapid estradiol-mediated enhancement of hippocampal synaptic transmission in mice.Differential action of monohydroxylated polycyclic aromatic hydrocarbons with estrogen receptors α and βThe role of estrogens in control of energy balance and glucose homeostasis.Interaction of 14-3-3 proteins with the estrogen receptor alpha F domain provides a drug target interface.Integrative genomics of gene and metabolic regulation by estrogen receptors α and β, and their coregulators.Agonist-mediated assembly of the crustacean methyl farnesoate receptor.Structurally similar estradiol analogs uniquely alter the regulation of intracellular signaling pathways.Monitoring Ligand-Activated Protein-Protein Interactions Using Bioluminescent Resonance Energy Transfer (BRET) Assay.Estrogen receptor beta2 and beta5 are associated with poor prognosis in prostate cancer, and promote cancer cell migration and invasion.Small-molecule hormones: molecular mechanisms of actionIn Situ Evaluation of Estrogen Receptor Dimers in Breast Carcinoma Cells: Visualization of Protein-Protein Interactions.Ligand-Mediated Receptor Assembly as an End Point for High-Throughput Chemical Toxicity Screening.Conservative nature of oestradiol signalling pathways in the brain lobes of octopus vulgaris involved in reproduction, learning and motor coordination.A computational based approach to identify estrogen receptor alpha/beta heterodimer selective ligands.Regulation of DNA Damage Response by Estrogen Receptor β-Mediated Inhibition of Breast Cancer Associated Gene 2.
P2860
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P2860
Intermolecular interactions identify ligand-selective activity of estrogen receptor alpha/beta dimers.
description
2008 nî lūn-bûn
@nan
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
2008年论文
@zh
2008年论文
@zh-cn
name
Intermolecular interactions id ...... en receptor alpha/beta dimers.
@en
type
label
Intermolecular interactions id ...... en receptor alpha/beta dimers.
@en
prefLabel
Intermolecular interactions id ...... en receptor alpha/beta dimers.
@en
P2860
P356
P1476
Intermolecular interactions id ...... en receptor alpha/beta dimers.
@en
P2093
P2860
P304
19012-19017
P356
10.1073/PNAS.0807274105
P407
P577
2008-11-20T00:00:00Z