Identification, synthesis and evaluation of substituted benzofurazans as inhibitors of CREB-mediated gene transcription. - Wikidata - wikimedia - TriplyDB

Identification, synthesis and evaluation of substituted benzofurazans as inhibitors of CREB-mediated gene transcription.

Identification, synthesis and evaluation of substituted benzofurazans as inhibitors of CREB-mediated gene transcription.

http://www.wikidata.org/entity/Q37198882

about

Control of CREB expression in tumors: from molecular mechanisms and signal transduction pathways to therapeutic target Novel Type of Prodrug Activation through a Long-Range O,N-Acyl Transfer: A Case of Water-Soluble CREB Inhibitor.PAINS in the assay: chemical mechanisms of assay interference and promiscuous enzymatic inhibition observed during a sulfhydryl-scavenging HTS.Identification of a Potent Inhibitor of CREB-Mediated Gene Transcription with Efficacious in Vivo Anticancer Activity.Irreversible binding of an anticancer compound (BI-94) to plasma proteins.Systemic Inhibition of CREB is Well-tolerated in vivo.Design, synthesis and biological evaluation of regioisomers of 666-15 as inhibitors of CREB-mediated gene transcription.Small molecule inhibition of cAMP response element binding protein in human acute myeloid leukemia cells.

P2860

Q28070887-749AC37D-A3F9-4299-BD8D-7549DE2F3776 Q34310220-46A6E2CA-466C-4B19-BB98-BA521BE59E63 Q34460371-057B8FA6-4492-42B2-9E5E-0AD82FB78984 Q35825716-99774D62-B178-44D3-82F7-CB88AD66C43D Q36005906-A4292180-C296-4168-8B64-5EF5E58C8F92 Q37303415-C4BFD8E3-BCCB-448C-94B5-131C9473993B Q38722053-CDA7C2FB-0387-406E-8870-8F9CA5AD3B42 Q38769308-B145701F-E6DB-4917-BB13-C53BA5D27DA0

P2860

Identification, synthesis and evaluation of substituted benzofurazans as inhibitors of CREB-mediated gene transcription.

http://www.wikidata.org/entity/Q37198882

description

article científic

@ca

article scientifique

@fr

articolo scientifico

@it

artigo científico

@pt

bilimsel makale

@tr

scientific article published on 31 July 2013

@en

vedecký článok

@sk

vetenskaplig artikel

@sv

videnskabelig artikel

@da

vědecký článek

@cs

name

Identification, synthesis and ...... B-mediated gene transcription.

@en

Identification, synthesis and ...... B-mediated gene transcription.

@nl

type

label

Identification, synthesis and ...... B-mediated gene transcription.

@en

Identification, synthesis and ...... B-mediated gene transcription.

@nl

prefLabel

Identification, synthesis and ...... B-mediated gene transcription.

@en

Identification, synthesis and ...... B-mediated gene transcription.

@nl

P1433

Q37198882-665D76CC-4AD8-4A06-B453-3D092673929F

P1476

Q37198882-F3D9DB00-F61B-4B88-9801-F7903F94F087

P2093

Q37198882-00DFB9EF-F300-4634-994A-4BD5396D0341

Q37198882-8B1DC854-769A-4D7E-8658-4AA7D7B94681

Q37198882-D89D9FE4-9D07-4788-BA37-383BEF1DF3A6

Q37198882-E7CF68AB-B9F2-4594-A2B0-14B2EB8A7E05

P2860

Q37198882-1286A95B-0315-4009-BDB2-D8C1445807D0

Q37198882-1E434507-D084-4C60-81F0-69319D773D1C

Q37198882-24554A27-4814-451E-A28A-A9FE6EFAF131

Q37198882-3A657620-14FC-4258-8B06-CD799154FFDE

Q37198882-4359D382-E7D2-40CC-A17B-0BAA3B8D3230

Q37198882-48AFA311-7BFE-4F57-B2F2-2CA7EFCD3FB3

Q37198882-540E4D36-90CA-41C5-A08F-001CEE37D243

Q37198882-541DFD0B-D4B0-48FC-9FE1-BB4FBDEECD7C

Q37198882-605A9E0C-C788-4F5E-A9A1-B3C989817915

Q37198882-605CE860-BCEB-48C7-A20D-61FC8E8B26D1

P304

Q37198882-21C0AD08-D0B4-41C2-9359-DA6485D8D4FE

P31

Q37198882-2B4C01A4-1855-41B7-A14B-6CB6DA470CBE

P356

Q37198882-EDFFBE81-609C-4344-B5EC-5CC4AD28B481

P407

Q37198882-5F845474-41C6-4CB1-873A-5DBE9B92EA2C

P433

Q37198882-8887F71C-8748-412D-9DAE-C53194F36304

P478

Q37198882-CC4703B7-C712-4751-911A-D84CEB11A691

P577

Q37198882-0BAF6D90-44D1-4769-BCA8-F56378D66E19

P5875

Q37198882-12971901-7321-446F-BF0E-96B8FA085959

P698

Q37198882-CF37F81E-F527-4E38-9826-52CA0E7FA45F

P932

Q37198882-DEC8C627-0993-4BD3-BCA4-073B9E1F35F6

P356

J.BMCL.2013.07.053

P1433

Bioorganic & Medicinal Chemistry Letters

P1476

Identification, synthesis and ...... B-mediated gene transcription.

@en

P2093

Bingbing X Li

http://www.w3.org/2001/XMLSchema#string

Candice Broussard

http://www.w3.org/2001/XMLSchema#string

Fuchun Xie

http://www.w3.org/2001/XMLSchema#string

Xiangshu Xiao

http://www.w3.org/2001/XMLSchema#string

P2860

P6981, An Arylstibonic Acid, Is a Novel Low Nanomolar Inhibitor of cAMP Response Element-Binding Protein Binding to DNA

Ordering a Dynamic Protein Via a Small-Molecule Stabilizer

Allosteric inhibition of hypoxia inducible factor-2 with small molecules

Solution Structure of the KIX Domain of CBP Bound to the Transactivation Domain of CREB: A Model for Activator:Coactivator Interactions

Transcriptional regulation by the phosphorylation-dependent factor CREB

Cyclic AMP stimulates somatostatin gene transcription by phosphorylation of CREB at serine 133

CREB: a stimulus-induced transcription factor activated by a diverse array of extracellular signals

Identification of small-molecule antagonists that inhibit an activator: coactivator interaction.

Design and synthesis of a cell-permeable synthetic transcription factor mimic.

Discovery of small molecule inhibitors of the PH domain leucine-rich repeat protein phosphatase (PHLPP) by chemical and virtual screening.

P304

5371-5375

http://www.w3.org/2001/XMLSchema#string

P31

scholarly article

P356

10.1016/J.BMCL.2013.07.053

http://www.w3.org/2001/XMLSchema#string

P407

P433

19

http://www.w3.org/2001/XMLSchema#string

P478

23

http://www.w3.org/2001/XMLSchema#string

P577

2013-07-31T00:00:00Z

http://www.w3.org/2001/XMLSchema#dateTime

P5875

255973575

http://www.w3.org/2001/XMLSchema#string

P698

23953193

http://www.w3.org/2001/XMLSchema#string

P932

3783659

http://www.w3.org/2001/XMLSchema#string