Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors

Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors

Item
http://www.wikidata.org/entity/Q37463122
Studying epigenetic complexes and their inhibitors with the proteomics toolboxEvolution of a Compact Photoprobe for the Dopamine Transporter Based on (±)-threo-Methylphenidate.On the inhibition of histone deacetylase 8Design, synthesis, modeling, biological evaluation and photoaffinity labeling studies of novel series of photoreactive benzamide probes for histone deacetylase 2.A One-Pot Selective Synthesis of N-Boc Protected Secondary Amines: Tandem Direct Reductive Amination/N-Boc Protection.Design, synthesis, docking, and biological evaluation of novel diazide-containing isoxazole- and pyrazole-based histone deacetylase probes.Novel histone deacetylase 8 ligands without a zinc chelating group: exploring an 'upside-down' binding pose.Insights from comprehensive multiple receptor docking to HDAC8.Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 5 Based on Select Acetylenic Negative Allosteric Modulators.Photoreactive "nanorulers" detect a novel conformation of full length HDAC3-SMRT complex in solutionRecent developments and applications of clickable photoprobes in medicinal chemistry and chemical biology.(±)-2-(N-tert-Butylamino)-3'-[(125)I]-iodo-4'-azidopropiophenone: a dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyban).Structure-activity relationships of hydroxamate-based histone deacetylase-8 inhibitors: reality behind anticancer drug discovery.Design, Synthesis, Molecular Modeling, and Biological Evaluation of Novel Amine-based Histone Deacetylase Inhibitors.Unambiguous Identification of β-Tubulin as the Direct Cellular Target Responsible for the Cytotoxicity of Chalcone by Photoaffinity Labeling.Design and development of histone deacetylase (HDAC) chemical probes for cell-based profiling.Magnetite nanoparticles coated with alkyne-containing polyacrylates for click chemistry
P2860

Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors

Item
http://www.wikidata.org/entity/Q37463122
description
2009 nî lūn-bûn
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2009年の論文
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2009年学术文章
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2009年学术文章
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2009年学术文章
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2009年学术文章
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2009年学术文章
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2009年學術文章
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name
Binding ensemble profiling wit ...... ding poses of HDAC8 inhibitors
@en
Binding ensemble profiling with photoaffinity labeling
@nl
type
label
Binding ensemble profiling wit ...... ding poses of HDAC8 inhibitors
@en
Binding ensemble profiling with photoaffinity labeling
@nl
prefLabel
Binding ensemble profiling wit ...... ding poses of HDAC8 inhibitors
@en
Binding ensemble profiling with photoaffinity labeling
@nl
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Binding ensemble profiling wit ...... ding poses of HDAC8 inhibitors
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P577
P5875
P698
P932