about
P300/CBP associated factor regulates nitroglycerin-dependent arterial relaxation by N(ε)-lysine acetylation of contractile proteinsAzole antifungal agents related to naftifine and butenafine.Small molecule inhibitors of histone arginine methyltransferases: homology modeling, molecular docking, binding mode analysis, and biological evaluations.Diversity through a branched reaction pathway: generation of multicyclic scaffolds and identification of antimigratory agents.Synthesis and evaluation of translocator 18 kDa protein (TSPO) positron emission tomography (PET) radioligands with low binding sensitivity to human single nucleotide polymorphism rs6971.Identification of small-molecule enhancers of arginine methylation catalyzed by coactivator-associated arginine methyltransferase 1.Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart.Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees.Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach.p300/CBP-associated factor selectively regulates the extinction of conditioned fear.Enhancement of lysine acetylation accelerates wound repair.Chemical biology of histone acetyltransferase natural compounds modulators.CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli.Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach.Identification of structural features of 2-alkylidene-1,3-dicarbonyl derivatives that induce inhibition and/or activation of histone acetyltransferases KAT3B/p300 and KAT2B/PCAF.Structure-activity relationship refinement and further assessment of 4-phenylquinazoline-2-carboxamide translocator protein ligands as antiproliferative agents in human glioblastoma tumors.Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells.Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors.Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.Modulation of the activity of histone acetyltransferases by long chain alkylidenemalonates (LoCAMs).Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1.Small-molecule inhibitors of protein geranylgeranyltransferase type I.6-alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): novel regulators of cell differentiation and proliferation.Synthesis and antifungal properties of N-[(1,1'-biphenyl)-4-ylmethyl]-1H-imidazol-1-amine derivatives.New structural analogues of Tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines.Synthesis and biochemical evaluation of δ(2)-isoxazoline derivatives as DNA methyltransferase 1 inhibitors.Synthesis of 3-aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole derivatives: a comparison between conventional, microwave-assisted and flow-based methodologies.Design, synthesis and biological evaluation of carboxy analogues of arginine methyltransferase inhibitor 1 (AMI-1).Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters.Antimycobacterial activity of ionic fullerene derivatives.A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines.Interaction of azole compounds with DOPC and DOPC/ergosterol bilayers by spin probe EPR spectroscopy: implications for antifungal activity.Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity.Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents.Effects of azole treatments on the physical properties of Candida albicans plasma membrane: a spin probe EPR study.Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes.Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases.Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases.
P50
Q28583676-40FF3BD4-F9DA-4667-8823-4761AFBD42E1Q31413042-1AFEA71A-2F6D-4C22-8ED7-E436BC52331DQ33275550-C5DD9AD8-E7D0-44A7-95C9-D243F051CC75Q33786011-F1D63631-565B-4CCB-AA2E-81751930A999Q34408079-AC80B4BB-2936-49CC-9BD6-2254E53967D9Q34456824-A6E81275-AB9F-48AD-BF22-D122070FDAE0Q34582749-E343ACC7-8BB9-488B-8F8A-ADC431186360Q34691702-4B305664-51F6-400C-B1FA-CFB86F9D9A1EQ36095575-09C31880-45C7-45DE-9468-A32740CACA27Q36303815-26ECB399-13C6-4CF4-B00E-AB71E3FFDDA0Q37313617-930B587A-94CC-419F-8B0F-65F955F3341AQ37825449-8942BBE9-E01C-4E09-BD3C-A5EDAE7107BCQ38867023-135D45D9-55EB-4EDA-B2E7-4BCBFC5B9A31Q38895557-E916E2F5-B4C5-4A7E-A00E-8E895A744211Q38904705-DA77E791-20FD-4649-8612-D256B160DBE5Q38946242-380E6D35-4D5E-4C36-BED2-FEFB01636F21Q39020023-E0FF5961-0C0D-4EB3-82F9-319A27A7F3ACQ39329294-5A4511AC-B359-4629-96D8-AB3205118345Q39366925-DAF4099D-1BA8-42EB-A4C2-27EFC3D10F13Q39506980-CCDA2356-30B4-49BF-9C20-40E538CD53D0Q39536678-42435C64-9465-4CF2-B746-B09123BA87E7Q39598116-18A8D06B-B22F-4409-9834-F52EBB815BD7Q40001720-ACEF609F-8E44-40B4-BC49-E594CB0DE156Q40144861-1BD35CA7-71AF-4E97-A30C-B51A290EDC61Q40237611-1A48002E-DC05-4ACA-A777-B17C9B0ABE0DQ40673323-4D7C7ACF-3B62-4703-98D1-C1067A65BF2CQ40835708-C5A9A482-B003-4C27-B70A-35405A595FBAQ42726505-29AE56E7-D160-486F-A80B-1A9119CD8396Q42873070-75CEDF52-7FCF-4CE0-8ADB-D6980D3C875EQ43187441-B8500CB2-AFE9-4F63-9352-ABEAF7BF6C3EQ43187779-9914D4D6-8F69-4AF9-B5B9-5A79EFB69408Q43503846-0C762093-C795-4332-9F42-4BAD2E60DA29Q43508487-67BD7428-5E14-4C4C-A7DE-3A02CEBBCBB0Q43738604-1725879D-5CD6-4870-BAAB-919920EA0F74Q43805720-0D192207-A8B8-4F78-B59A-6229E4533AADQ44522237-CC2CC948-7250-436E-BF96-BB4D8A04E954Q44689079-D1271B23-3E87-40D7-ABAE-675B4757AE1EQ45414691-78A7A867-A5A4-4F20-A114-21EA32444C92Q46162765-8CC7DA9F-F713-407C-BB7A-7E701285C169Q46628836-8BC8B576-A66A-4D66-A242-2A0BC1EA0769
P50
description
hulumtuese
@sq
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Sabrina Castellano
@ast
Sabrina Castellano
@en
Sabrina Castellano
@es
Sabrina Castellano
@nl
Sabrina Castellano
@sl
type
label
Sabrina Castellano
@ast
Sabrina Castellano
@en
Sabrina Castellano
@es
Sabrina Castellano
@nl
Sabrina Castellano
@sl
prefLabel
Sabrina Castellano
@ast
Sabrina Castellano
@en
Sabrina Castellano
@es
Sabrina Castellano
@nl
Sabrina Castellano
@sl
P106
P1153
7004170198
P21
P31
P496
0000-0002-7449-3704