6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
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Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitors.Modulation of HIV-1-induced activation of plasmacytoid dendritic cells by 6-desfluoroquinolones.Strategies to Block HIV Transcription: Focus on Small Molecule Tat Inhibitors.Targeting HIV transcription: the quest for a functional cure.Recent advances in the identification of Tat-mediated transactivation inhibitors: progressing toward a functional cure of HIV.A new vinyl selenone-based domino approach to spirocyclopropyl oxindoles endowed with anti-HIV RT activity.Tumour cell population growth inhibition and cell death induction of functionalized 6-aminoquinolone derivatives.Computer-aided design, synthesis and validation of 2-phenylquinazolinone fragments as CDK9 inhibitors with anti-HIV-1 Tat-mediated transcription activity.Design, synthesis, and evaluation of WC5 analogues as inhibitors of human cytomegalovirus Immediate-Early 2 protein, a promising target for anti-HCMV treatment.Chiral separation of quinolones by liquid chromatography and capillary electrophoresis.Structural investigation of the naphthyridone scaffold: identification of a 1,6-naphthyridone derivative with potent and selective anti-HIV activity.From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors
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P2860
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
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article científic
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article scientifique
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articolo scientifico
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artigo científico
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bilimsel makale
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scientific article published on July 2010
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vedecký článok
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vetenskaplig artikel
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videnskabelig artikel
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vědecký článek
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name
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
@en
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
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type
label
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
@en
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
@nl
prefLabel
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
@en
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors.
@nl
P2093
P2860
P50
P356
P1476
6-desfluoroquinolones as HIV-1 Tat-mediated transcription inhibitors
@en
P2093
Oriana Tabarrini
Serena Massari
Violetta Cecchetti
P2860
P304
P356
10.4155/FMC.10.208
P577
2010-07-01T00:00:00Z