Allosteric modulators of rhodopsin-like G protein-coupled receptors: opportunities in drug development.
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Identification of G protein-coupled receptors in Schistosoma haematobium and S. mansoni by comparative genomics.Role of G-protein-coupled receptor-related genes in insecticide resistance of the mosquito, Culex quinquefasciatusMedicinal chemistry of adenosine, P2Y and P2X receptors.Computational Tools for Allosteric Drug Discovery: Site Identification and Focus Library Design.Bioinformatic prediction of G protein-coupled receptor encoding sequences from the transcriptome of the foreleg, including the Haller's organ, of the cattle tick, Rhipicephalus australis.ASD v3.0: unraveling allosteric regulation with structural mechanisms and biological networks.GPCR and IR genes in Schistosoma mansoni miracidiaStructure-activity relationship study of indole-2-carboxamides identifies a potent allosteric modulator for the cannabinoid receptor 1 (CB1).Harnessing allostery: a novel approach to drug discovery.Allosteric Inhibition of Serotonin 5-HT7 Receptors by Zinc Ions.Pyrimidinyl Biphenylureas: Identification of New Lead Compounds as Allosteric Modulators of the Cannabinoid Receptor CB1.Synthesis and biological evaluation of indole-2-carboxamides bearing photoactivatable functionalities as novel allosteric modulators for the cannabinoid CB1 receptor.Detection and quantification of allosteric modulation of endogenous m4 muscarinic acetylcholine receptor using impedance-based label-free technology in a neuronal cell line.The cell biology of the thyroid-disrupting mechanism of dichlorodiphenyltrichloroethane (DDT).Development of [(3)H]2-Carboxy-4,6-dichloro-1H-indole-3-propionic Acid ([(3)H]PSB-12150): A Useful Tool for Studying GPR17Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor.The rat adenine receptor: pharmacological characterization and mutagenesis studies to investigate its putative ligand binding site.New pipelines for novel allosteric GPCR modulatorsAnalysis of Pelagia noctiluca proteome Reveals a Red Fluorescent Protein, a Zinc Metalloproteinase and a Peroxiredoxin.Opportunities and Challenges in the Discovery of Allosteric Modulators of GPCRs.
P2860
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P2860
Allosteric modulators of rhodopsin-like G protein-coupled receptors: opportunities in drug development.
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article científic
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article scientifique
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articol științific
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articolo scientifico
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artigo científico
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artigo científico
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artigo científico
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artikel ilmiah
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artikull shkencor
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artículo científico
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name
Allosteric modulators of rhodo ...... rtunities in drug development.
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type
label
Allosteric modulators of rhodo ...... rtunities in drug development.
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prefLabel
Allosteric modulators of rhodo ...... rtunities in drug development.
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P50
P1476
Allosteric modulators of rhodo ...... rtunities in drug development.
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P304
P356
10.1016/J.PHARMTHERA.2012.06.002
P577
2012-06-19T00:00:00Z