Small-molecule inhibitors binding to protein kinases. Part I: exceptions from the traditional pharmacophore approach of type I inhibition.
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SD-208, a novel protein kinase D inhibitor, blocks prostate cancer cell proliferation and tumor growth in vivo by inducing G2/M cell cycle arrestKinetic capillary electrophoresis with mass-spectrometry detection (KCE-MS) facilitates label-free solution-based kinetic analysis of protein-small molecule binding.Small molecule c-Met kinase inhibitors: a review of recent patents.Design, synthesis and evaluation of 2-phenylisothiazolidin-3-one-1,1-dioxides as a new class of human protein kinase CK2 inhibitors.Targeting the DFG-in kinase conformation: a new trend emerging from a patent analysis.p38α mitogen-activated protein kinase inhibitors, a patent review (2005-2011).Synthesis and p38 Inhibitory Activity of Some Novel Substituted N,N'-Diarylurea Derivatives.Identification of novel inhibitors for Pim-1 kinase using pharmacophore modeling based on a novel method for selecting pharmacophore generation subsets.Design, synthesis and biological evaluation of 2-aminopyrimidinones and their 6-aza-analogs as a new class of CK2 inhibitors.Application of shape-based and pharmacophore-based in silico screens for identification of Type II protein kinase inhibitors.
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Small-molecule inhibitors binding to protein kinases. Part I: exceptions from the traditional pharmacophore approach of type I inhibition.
description
article científic
@ca
article scientifique
@fr
articol științific
@ro
articolo scientifico
@it
artigo científico
@gl
artigo científico
@pt
artigo científico
@pt-br
artikel ilmiah
@id
artikull shkencor
@sq
artículo científico
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name
Small-molecule inhibitors bind ...... approach of type I inhibition.
@en
type
label
Small-molecule inhibitors bind ...... approach of type I inhibition.
@en
prefLabel
Small-molecule inhibitors bind ...... approach of type I inhibition.
@en
P2093
P2860
P1476
Small-molecule inhibitors bind ...... approach of type I inhibition.
@en
P2093
P2860
P304
P356
10.1517/17460440802579975
P407
P577
2008-12-01T00:00:00Z