about
Discovery of a new efficient chiral ligand for copper-catalyzed enantioselective Michael additions by high-throughput screening of a parallel library.Rh-catalyzed asymmetric hydrogenation of prochiral olefins with a dynamic library of chiral TROPOS phosphorus ligands.Bicyclic carbohydrate-derived scaffolds for combinatorial libraries.Rh-catalyzed enantioselective conjugate addition of arylboronic acids with a dynamic library of chiral tropos phosphorus ligands.Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF ReceptorsInsights into the Binding of Cyclic RGD Peptidomimetics to α5β1 Integrin by using Live-Cell NMR And Computational Studies.αvβ3 Integrin-Targeted Peptide/Peptidomimetic-Drug Conjugates: In-Depth Analysis of the Linker Technology.Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers.Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonists.Synthesis and biological evaluation of dual action cyclo-RGD/SMAC mimetic conjugates targeting α(v)β(3)/α(v)β(5) integrins and IAP proteins.Determination of the binding epitope of RGD-peptidomimetics to αvβ3 and α(IIb)β3 integrin-rich intact cells by NMR and computational studies.Tumor Targeting with an isoDGR-Drug Conjugate2,3-Dihydroxybenzoate pathway in Pseudomonas putida. 1H n.m.r. study on the ring-cleavage site.Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αV β3.Cyclic RGD-peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands.Cyclic isoDGR peptidomimetics as low-nanomolar αvβ3 integrin ligands.A straightforward total synthesis of (-)-chaetominine.A formal total synthesis of eleutherobin using the ring-closing metathesis (RCM) reaction of a densely functionalized diene as the key step: investigation of the unusual kinetically controlled RCM stereochemistry.Enantioselective conjugate addition of phenylboronic acid to enones catalysed by a chiral tropos/atropos rhodium complex at the coalescence temperature.Synthesis and conformational studies of peptidomimetics containing a new bifunctional diketopiperazine scaffold acting as a beta-hairpin inducer.A practical approach to the resolution of racemic N-benzyl alpha-amino acids by liquid-liquid extraction with a lipophilic chiral salen-cobalt(III) complex.Investigating the Interaction of Cyclic RGD Peptidomimetics with αVβ₆ Integrin by Biochemical and Molecular Docking Studies.Efficient resolution of racemic N-benzyl beta3-amino acids by iterative liquid-liquid extraction with a chiral (salen)cobalt(III) complex as enantioselective selector.Supramolecular ligand-ligand and ligand-substrate interactions for highly selective transition metal catalysis.Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting.Enantioselective binding of dipeptides using acyclic receptorsSynthesis, Conformational Studies and Binding Properties of Acyclic Receptors for N-Protected Amino Acids and DipeptidesLewis acid mediated aldol condensations using thioester silyl ketene acetalsTheoretical studies of stereoselective aldol condensationsImproving C=N Bond Reductions with (Cyclopentadienone)iron Complexes: Scope and LimitationsFrontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αV β3Riding the Wave of Monodentate Ligand Revival: From the A/B Concept to Noncovalent InteractionsAsymmetric Hydrogenation of 3-Substituted Pyridinium SaltsCyclic RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin LigandsPhthalaPhos: Chiral Supramolecular Ligands for Enantioselective Rhodium-Catalyzed Hydrogenation ReactionsCombination of a binaphthol-derived phosphite and a C1-symmetric phosphinamine generates heteroleptic catalysts in Rh- and Pd-mediated reactionsA highly stereoselective synthesis of the C10–C23 fragment of (–)-dictyostatinA Formal Total Synthesis of Eleutherobin Through an Unprecedented Kinetically Controlled Ring-Closing-Metathesis Reaction of a Densely Functionalized DieneCopper catalysed 1,4-addition of organozinc reagents to α,β-unsaturated carbonyl compounds: a mechanistic investigationCopper Phosphoramidite-Catalyzed Enantioselective Desymmetrization of meso-Cyclic Allylic Bisdiethyl Phosphates
P50
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P50
description
hulumtues
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researcher
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wetenschapper
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հետազոտող
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name
Cesare Gennari
@ast
Cesare Gennari
@en
Cesare Gennari
@es
Cesare Gennari
@nl
Cesare Gennari
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type
label
Cesare Gennari
@ast
Cesare Gennari
@en
Cesare Gennari
@es
Cesare Gennari
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Cesare Gennari
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prefLabel
Cesare Gennari
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Cesare Gennari
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Cesare Gennari
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Cesare Gennari
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Cesare Gennari
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P1053
P-4430-2016
P106
P1153
7102020772
P21
P31
P3829
P496
0000-0002-7635-4900