about
X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitutionCharacterization of HIV-1 resistance to a fusion inhibitor, N36, derived from the gp41 amino-terminal heptad repeatStructure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitorsIdentification of novel low molecular weight CXCR4 antagonists by structural tuning of cyclic tetrapeptide scaffolds.Molecular-size reduction of a potent CXCR4-chemokine antagonist using orthogonal combination of conformation- and sequence-based libraries.Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: disclosing the importance of side-chain and backbone functionalities.Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the phosphotyrosyl+1 position of Grb2 SH2 domain-binding tripeptides.Structure-activity relationship study on polyglutamine binding peptide QBP1.Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids.Activation of Neuropeptide FF Receptors by Kisspeptin Receptor Ligands.A potent chemotherapeutic strategy for bladder cancer: (S)-methoxy-trityl-L-cystein, a novel Eg5 inhibitor.A potent chemotherapeutic strategy in prostate cancer: S-(methoxytrityl)-L-cysteine, a novel Eg5 inhibitorMechanism of resistance to S138A substituted enfuvirtide and its application to peptide designMolecular modeling study of cyclic pentapeptide CXCR4 antagonists: new insight into CXCR4-FC131 interactions.Rapid mobilization of hematopoietic progenitors by AMD3100 and catecholamines is mediated by CXCR4-dependent SDF-1 release from bone marrow stromal cells.Stromal cell-derived factor 1 regulates the actin organization of chondrocytes and chondrocyte hypertrophyResistance profiles of novel electrostatically constrained HIV-1 fusion inhibitors.Optimized method of G-protein-coupled receptor homology modeling: its application to the discovery of novel CXCR7 ligands.Kisspeptin neurons mediate reflex ovulation in the musk shrew (Suncus murinus)A HAMP promoter bioassay system for identifying chemical compounds that modulate hepcidin expression.Design, synthesis, and structure-activity relationships of 1-ethylpyrazole-3-carboxamide compounds as novel hypoxia-inducible factor (HIF)-1 inhibitors.Structure-activity relationship studies on cyclic RGD peptides utilizing novel alkene dipeptide isosteres.Screening of a virtual mirror-image library of natural products.Potent anti-HIV-1 activity of N-HR-derived peptides including a deep pocket-forming region without antagonistic effects on T-20GnRH suppresses excitability of visual processing neurons in the optic tectum.Plasmodium falciparum domain mediating adhesion to chondroitin sulfate A: a receptor for human placental infection.Therapeutic potential of the chemokine receptor CXCR4 antagonists as multifunctional agents.HIV-1 resistance mechanism to an electrostatically constrained peptide fusion inhibitor that is active against T-20-resistant strainsDesign of peptide-based inhibitors for human immunodeficiency virus type 1 strains resistant to T-20SC29EK, a peptide fusion inhibitor with enhanced alpha-helicity, inhibits replication of human immunodeficiency virus type 1 mutants resistant to enfuvirtidePeptide and peptidomimetic ligands for CXC chemokine receptor 4 (CXCR4).Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction.Impact of HIV-1 infection pathways on susceptibility to antiviral drugs and on virus spread.Neuropeptide derivatives to regulate the reproductive axis: Kisspeptin receptor (KISS1R) ligands and neurokinin-3 receptor (NK3R) ligands.Potential new chemotherapy strategy for human ovarian carcinoma with a novel KSP inhibitor.Synthesis of IB-01212 by multiple N-methylations of peptide bonds.Polyamine modification by acrolein exclusively produces 1,5-diazacyclooctanes: a previously unrecognized mechanism for acrolein-mediated oxidative stress.Design and synthesis of fluorescent probes for GPR54.A simple, rapid, and sensitive system for the evaluation of anti-viral drugs in rats.Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182.
P50
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P50
description
hulumtues
@sq
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Shinya Oishi
@ast
Shinya Oishi
@en
Shinya Oishi
@es
Shinya Oishi
@nl
Shinya Oishi
@sl
type
label
Shinya Oishi
@ast
Shinya Oishi
@en
Shinya Oishi
@es
Shinya Oishi
@nl
Shinya Oishi
@sl
prefLabel
Shinya Oishi
@ast
Shinya Oishi
@en
Shinya Oishi
@es
Shinya Oishi
@nl
Shinya Oishi
@sl
P1053
C-1350-2011
P106
P21
P31
P3829
P496
0000-0002-2833-2539