Trace amine-associated receptor 1 displays species-dependent stereoselectivity for isomers of methamphetamine, amphetamine, and para-hydroxyamphetamine.
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Trace amine-associated receptors as emerging therapeutic targetsThe emerging role of trace amine-associated receptor 1 in the functional regulation of monoamine transporters and dopaminergic activityTrace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine classPharmacological characterization of membrane-expressed human trace amine-associated receptor 1 (TAAR1) by a bioluminescence resonance energy transfer cAMP biosensorInternational Union of Pharmacology. LXXII. Recommendations for trace amine receptor nomenclatureA receptor mechanism for methamphetamine action in dopamine transporter regulation in brainTrace amine-associated receptor 1-Family archetype or iconoclast?Trace amine-associated receptor 1 as a monoaminergic modulator in brainTrace Amines and the Trace Amine-Associated Receptor 1: Pharmacology, Neurochemistry, and Clinical ImplicationsRactopamine, a livestock feed additive, is a full agonist at trace amine-associated receptor 1"TAARgeting Addiction"--The Alamo Bears Witness to Another Revolution: An Overview of the Plenary Symposium of the 2015 Behavior, Biology and Chemistry ConferenceDeterminants involved in subtype-specific functions of rat trace amine-associated receptors 1 and 4Pharmacotherapeutic agents in the treatment of methamphetamine dependence.Functional evolution of the trace amine associated receptors in mammals and the loss of TAAR1 in dogs.Structural and functional evolution of the trace amine-associated receptors TAAR3, TAAR4 and TAAR5 in primates.Genetic Polymorphisms Affect Mouse and Human Trace Amine-Associated Receptor 1 Function.Interactions of HIV and drugs of abuse: the importance of glia, neural progenitors, and host genetic factors.Augmentation of methamphetamine-induced behaviors in transgenic mice lacking the trace amine-associated receptor 1Trace amine-associated receptor 1 (TAAR1) is activated by amiodarone metabolitesAvenues for the development of therapeutics that target trace amine associated receptor 1 (TAAR1).Cloning, expression, and functional analysis of rhesus monkey trace amine-associated receptor 6: evidence for lack of monoaminergic association.The molecular basis of species-specific ligand activation of trace amine-associated receptor 1 (TAAR(1)).Structure-activity correlations for beta-phenethylamines at human trace amine receptor 1.The trace amine-associated receptor 1 modulates methamphetamine's neurochemical and behavioral effects.Evolutionary Conservation of 3-Iodothyronamine as an Agonist at the Trace Amine-Associated Receptor 1.Trace Amine-Associated Receptor 1 Localization at the Apical Plasma Membrane Domain of Fisher Rat Thyroid Epithelial Cells Is Confined to Cilia.In Vitro Characterization of Psychoactive Substances at Rat, Mouse, and Human Trace Amine-Associated Receptor 1.A partial trace amine-associated receptor 1 agonist exhibits properties consistent with a methamphetamine substitution treatment.The Case for TAAR1 as a Modulator of Central Nervous System Function.Trace amine-associated receptors can bind trace aminesTAAR1 in Addiction: Looking Beyond the Tip of the Iceberg.
P2860
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P2860
Trace amine-associated receptor 1 displays species-dependent stereoselectivity for isomers of methamphetamine, amphetamine, and para-hydroxyamphetamine.
description
2007 nî lūn-bûn
@nan
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
2007年论文
@zh
2007年论文
@zh-cn
name
Trace amine-associated recepto ...... , and para-hydroxyamphetamine.
@en
type
label
Trace amine-associated recepto ...... , and para-hydroxyamphetamine.
@en
prefLabel
Trace amine-associated recepto ...... , and para-hydroxyamphetamine.
@en
P2093
P356
P1476
Trace amine-associated recepto ...... , and para-hydroxyamphetamine.
@en
P2093
Arttamangkul S
Sonders MS
P304
P356
10.1124/JPET.106.115402
P407
P577
2007-01-11T00:00:00Z