Differential helical orientations among related G protein-coupled receptors provide a novel mechanism for selectivity. Studies with salvinorin A and the kappa-opioid receptor.
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Structure of the human κ-opioid receptor in complex with JDTicKappa opioids promote the proliferation of astrocytes via Gbetagamma and beta-arrestin 2-dependent MAPK-mediated pathwaysStructure-based design, synthesis, and biochemical and pharmacological characterization of novel salvinorin A analogues as active state probes of the kappa-opioid receptorHerkinorin analogues with differential beta-arrestin-2 interactionsSingle Amino Acid Variation Underlies Species-Specific Sensitivity to Amphibian Skin-Derived Opioid-like Peptides.FoldGPCR: structure prediction protocol for the transmembrane domain of G protein-coupled receptors from class A.Salvinorin A analogs as probes in opioid pharmacology.Neuropharmacology of the naturally occurring kappa-opioid hallucinogen salvinorin ACoMFA analyses of C-2 position salvinorin A analogs at the kappa-opioid receptor provides insights into epimer selectivity.Synthetic studies of neoclerodane diterpenes from Salvia divinorum: role of the furan in affinity for opioid receptorsOpioid receptor probes derived from cycloaddition of the hallucinogen natural product salvinorin A.Utilizing nature as a source of new probes for opioid pharmacology.Allosteric modulation model of the mu opioid receptor by herkinorin, a potent not alkaloidal agonist.Modular Approach to pseudo-Neoclerodanes as Designer κ-Opioid Ligands.
P2860
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P2860
Differential helical orientations among related G protein-coupled receptors provide a novel mechanism for selectivity. Studies with salvinorin A and the kappa-opioid receptor.
description
2006 nî lūn-bûn
@nan
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
2006年论文
@zh
2006年论文
@zh-cn
name
Differential helical orientati ...... and the kappa-opioid receptor.
@en
type
label
Differential helical orientati ...... and the kappa-opioid receptor.
@en
prefLabel
Differential helical orientati ...... and the kappa-opioid receptor.
@en
P2093
P2860
P356
P1476
Differential helical orientati ...... and the kappa-opioid receptor.
@en
P2093
Bryan L Roth
Philip D Mosier
Richard B Westkaemper
Timothy A Vortherms
P2860
P304
P356
10.1074/JBC.M609264200
P407
P577
2006-11-22T00:00:00Z