Unsulfated C-terminal 7-peptide of cholecystokinin: a new ligand of the opiate receptor.
about
Type and location of fluorescent probes incorporated into the potent mu-opioid peptide [Dmt]DALDA affect potency, receptor selectivity and intrinsic efficacy."Carba"-analogues of fentanyl are opioid receptor agonists.Cyclic enkephalin-deltorphin hybrids containing a carbonyl bridge: structure and opioid activity.'Carba'-carfentanil (trans isomer): a μ opioid receptor (MOR) partial agonist with a distinct binding mode.N-methylated cyclic enkephalin analogues retain high opioid receptor binding affinity.Bifunctional μ/δ opioid peptides: variation of the type and length of the linker connecting the two componentsA cyclic enkephalin analog with high in vitro opiate activity.Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries.Dicarba analogues of the cyclic enkephalin peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) retain high opioid activityCyclic opioid peptide agonists and antagonists obtained via ring-closing metathesis.A Cyclic Tetrapeptide ("Cyclodal") and Its Mirror-Image Isomer Are Both High-Affinity μ Opioid Receptor Antagonists.Cyclic enkephalins with a diversely substituted guanidine bridge or a thiourea bridge: synthesis, biological and structural evaluations.[Dmt(1)]DALDA analogues with enhanced μ opioid agonist potency and with a mixed μ/κ opioid activity profileYFa and analogs: investigation of opioid receptors in smooth muscle contraction.Opiate antagonistic function of cholecystokinin in analgesia and energy balance systems.Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice.Variation of the net charge, lipophilicity, and side chain flexibility in Dmt(1)-DALDA: Effect on Opioid Activity and Biodistribution.Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 receptor antagonist.Highly potent side-chain to side-chain cyclized enkephalin analogues containing a carbonyl bridge: synthesis, biology and conformation.A chimeric opioid peptide with mixed mu agonist/delta antagonist properties.
P2860
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P2860
Unsulfated C-terminal 7-peptide of cholecystokinin: a new ligand of the opiate receptor.
description
1978 nî lūn-bûn
@nan
1978年の論文
@ja
1978年論文
@yue
1978年論文
@zh-hant
1978年論文
@zh-hk
1978年論文
@zh-mo
1978年論文
@zh-tw
1978年论文
@wuu
1978年论文
@zh
1978年论文
@zh-cn
name
Unsulfated C-terminal 7-peptide of cholecystokinin: a new ligand of the opiate receptor.
@en
type
label
Unsulfated C-terminal 7-peptide of cholecystokinin: a new ligand of the opiate receptor.
@en
prefLabel
Unsulfated C-terminal 7-peptide of cholecystokinin: a new ligand of the opiate receptor.
@en
P2093
P1476
Unsulfated C-terminal 7-peptide of cholecystokinin: a new ligand of the opiate receptor.
@en
P2093
Bodanszky M
Horrobin DF
Schiller PW
P304
P356
10.1016/0006-291X(78)91149-X
P577
1978-12-01T00:00:00Z