Synthesis and evaluation of 4-substituted piperidines and piperazines as balanced affinity μ opioid receptor (MOR) agonist/δ opioid receptor (DOR) antagonist ligands.
about
Further Optimization and Evaluation of Bioavailable, Mixed-Efficacy μ-Opioid Receptor (MOR) Agonists/δ-Opioid Receptor (DOR) Antagonists: Balancing MOR and DOR Affinities.Molecular Pharmacology of δ-Opioid Receptors.Asymmetric synthesis and in vitro and in vivo activity of tetrahydroquinolines featuring a diverse set of polar substitutions at the 6 position as mixed-efficacy μ opioid receptor/δ opioid receptor ligands.Crystal structures of 4-phenyl-piperazin-1-ium 6-chloro-5-ethyl-2,4-dioxopyrimidin-1-ide and 4-phenyl-piperazin-1-ium 6-chloro-5-isopropyl-2,4-dioxopyrimidin-1-ide.Rapid Synthesis of Boc-2',6'-dimethyl-l-tyrosine and Derivatives and Incorporation into Opioid Peptidomimetics.
P2860
Synthesis and evaluation of 4-substituted piperidines and piperazines as balanced affinity μ opioid receptor (MOR) agonist/δ opioid receptor (DOR) antagonist ligands.
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
2013年论文
@zh
2013年论文
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name
Synthesis and evaluation of 4- ...... ptor (DOR) antagonist ligands.
@en
type
label
Synthesis and evaluation of 4- ...... ptor (DOR) antagonist ligands.
@en
prefLabel
Synthesis and evaluation of 4- ...... ptor (DOR) antagonist ligands.
@en
P2093
P2860
P1476
Synthesis and evaluation of 4- ...... ptor (DOR) antagonist ligands.
@en
P2093
Aaron M Bender
Henry I Mosberg
John R Traynor
Mary J Clark
Michael P Agius
P2860
P304
P356
10.1016/J.BMCL.2013.12.021
P407
P577
2013-12-11T00:00:00Z