Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR
about
The role of brain somatostatin receptor 2 in the regulation of feeding and drinking behaviorPattern of Fos expression in the brain induced by selective activation of somatostatin receptor 2 in ratsBrain somatostatin receptor 2 mediates the dipsogenic effect of central somatostatin and cortistatin in rats: role in drinking behavior.Abdominal surgery inhibits circulating acyl ghrelin and ghrelin-O-acyltransferase levels in rats: role of the somatostatin receptor subtype 2.Selective agonists of somatostatin receptor subtype 1 or 2 injected peripherally induce antihyperalgesic effect in two models of visceral hypersensitivity in miceModulation of the adaptive response to stress by brain activation of selective somatostatin receptor subtypes.Novel, potent, and radio-iodinatable somatostatin receptor 1 (sst1) selective analoguesAnticonvulsant neuropeptides as drug leads for neurological diseases.Improvement of drug-like properties of peptides: the somatostatin paradigm.Central actions of somatostatin-28 and oligosomatostatin agonists to prevent components of the endocrine, autonomic and visceral responses to stress through interaction with different somatostatin receptor subtypes.In vitro structure-activity relationship of Re-cyclized octreotide analogues.Design and in vitro characterization of highly sst2-selective somatostatin antagonists suitable for radiotargeting.Ring size in octreotide amide modulates differently agonist versus antagonist binding affinity and selectivity.Selective central activation of somatostatin receptor 2 increases food intake, grooming behavior and rectal temperature in rats.Activation of brain somatostatin 2 receptors stimulates feeding in mice: analysis of food intake microstructure.Central somatostatin receptor 1 activation reverses acute stress-related alterations of gastric and colonic motor function in micePeptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine.DOTA-Derivatives of Octreotide Dicarba-Analogs with High Affinity for Somatostatin sst2,5 Receptors.Activation of somatostatin 2 receptors in the brain and the periphery induces opposite changes in circulating ghrelin levels: functional implications.Ring size of somatostatin analogues (ODT-8) modulates receptor selectivity and binding affinity.Central administration of pan-somatostatin agonist ODT8-SST prevents abdominal surgery-induced inhibition of circulating ghrelin, food intake and gastric emptying in rats.Three-dimensional consensus structure of sst2-selective somatostatin (SRIF) antagonists by NMR.Insights into structure-activity relationships of somatostatin analogs containing mesitylalanine.Fine-tuning the π-π aromatic interactions in peptides: somatostatin analogues containing mesityl alanine.
P2860
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P2860
Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR
description
2006 nî lūn-bûn
@nan
2006年の論文
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2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
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2006年论文
@wuu
2006年论文
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2006年论文
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name
Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR
@en
type
label
Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR
@en
prefLabel
Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR
@en
P2093
P2860
P356
P1476
Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR
@en
P2093
Christy Rani R Grace
Jean Rivier
Judit Erchegyi
Roland Riek
Steven C Koerber
P2860
P304
P356
10.1021/JM060363V
P407
P577
2006-07-01T00:00:00Z