Studies on RX 781094: a selective, potent and specific antagonist of alpha 2-adrenoceptors.
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The pharmacology of fluparoxan: a selective alpha 2-adrenoceptor antagonistA comparative study of the reversal by different alpha 2-adrenoceptor antagonists of the central sympatho-inhibitory effect of clonidineMediation of the antidepressant-like effect of 8-OH-DPAT in mice by postsynaptic 5-HT1A receptorsEvidence for a peripheral component in the sympatholytic effect of clonidine in ratsPharmacological effects and pharmacokinetics of atipamezole, a novel alpha 2-adrenoceptor antagonist--a randomized, double-blind cross-over study in healthy male volunteersAdrenergic receptors modulate motoneuron excitability, sensory synaptic transmission and muscle spasms after chronic spinal cord injury.α(2A) adrenergic receptor promotes amyloidogenesis through disrupting APP-SorLA interactionContribution of alpha-adrenoceptors to depolarization and contraction evoked by continuous asynchronous sympathetic nerve activity in rat tail artery.Attenuation of tolerance to opioid-induced antinociception and protection against morphine-induced decrease of neurofilament proteins by idazoxan and other I2-imidazoline ligands.Effects of idazoxan on alcohol pharmacokinetics and intoxication: a preliminary human laboratory study.Roles of serotonergic and adrenergic receptors in the antinociception of selective cyclooxygenase-2 inhibitor in the rat spinal cordModulation of the actions of tyrosine by alpha 2-adrenoceptor blockade.The thermogenic actions of alpha 2-adrenoceptor agonists in reserpinized mice are mediated via a central postsynaptic alpha 2-adrenoceptor mechanism.Alpha 2-adrenoceptor agonists enhance vasoconstrictor responses to alpha 1-adrenoceptor agonists in the rat tail artery by increasing the influx of Ca2+.Imidazoline binding sites in human placenta: evidence for heterogeneity and a search for physiological function[3H]-rauwolscine binding to alpha 2-adrenoceptors in the mammalian kidney: apparent receptor heterogeneity between species.Evidence for autoinhibition of stimulation-induced noradrenaline release from vasa deferentia of the guinea-pig and rat.Suppression by neuropeptide Y of capsaicin-sensitive sensory nerve-mediated contraction in guinea-pig airways.Effects of reduced calcium ion concentration and of diltiazem on vasoconstrictor responses to noradrenaline and sympathetic nerve stimulation in rat isolated tail artery.Pharmacological activity of ACC-7513, a selective alpha-adrenoceptor and 5-hydroxytryptamine receptor blocking agentInteraction between the inhibitory action of acetylcholine and the alpha-adrenoceptor autoinhibitory feedback system on release of [3H]-noradrenaline from rat atria and rabbit ear arteryThe alpha2 adrenergic receptor antagonist idazoxan, but not the serotonin-2A receptor antagonist M100907, partially attenuated reward deficits associated with nicotine, but not amphetamine, withdrawal in ratsActivation of sympathetic nerves exerts an inhibitory influence on afferent nerve-induced vasodilation unrelated to vasoconstriction in rat dental pulp.Alpha-adrenoceptors: a critical review.Localization of I2-imidazoline binding sites on monoamine oxidases.Compounds acting on alpha 1- and alpha 2- adrenoceptors: agonists and antagonists.Receptor-receptor interactions in the central nervous system. A new integrative mechanism in synapses.Role of imidazoline receptors in halothane-epinephrine arrhythmias.Alpha 2-adrenergic hyperpolarization is not involved in slow synaptic inhibition in amphibian sympathetic ganglia.Neuronal responses to noradrenaline in the cerebral cortex: evidence against the involvement of alpha 2-adrenoceptors.The role of alpha-adrenoceptors in the regulation of renal tubular sodium reabsorption and renin secretion in the rabbit.2-Alkyl analogue of idazoxan (RX 781094) with enhanced antagonist potency and selectivity at central alpha 2-adrenoceptors in the ratSelectivity and potency of 2-alkyl analogues of the alpha 2-adrenoceptor antagonist idazoxan (RX 781094) in peripheral systems.Activation and desensitization of presynaptic alpha 2-adrenoceptors after inhibition of neuronal uptake by antidepressant drugs in the rat vas deferens.The effect of alpha 2-adrenoceptor agonists on the acid secretory responses of rat isolated gastric mucosa to electrical field stimulation.[3H]-RS-15385-197, a selective and high affinity radioligand for alpha 2-adrenoceptors: implications for receptor classification.Noradrenaline-induced constriction of large and small coronary arteries in the anaesthetized dog.Characterization and autoradiographical localization of non-adrenoceptor idazoxan binding sites in the rat brain.The physiological and pharmacological role of presynaptic alpha- and beta-adrenoceptors in man.Adaptive changes in alpha-2 adrenoceptor mediated responses: analgesia, hypothermia and hypoactivity.
P2860
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P2860
Studies on RX 781094: a selective, potent and specific antagonist of alpha 2-adrenoceptors.
description
1983 nî lūn-bûn
@nan
1983年の論文
@ja
1983年論文
@yue
1983年論文
@zh-hant
1983年論文
@zh-hk
1983年論文
@zh-mo
1983年論文
@zh-tw
1983年论文
@wuu
1983年论文
@zh
1983年论文
@zh-cn
name
Studies on RX 781094: a select ...... nist of alpha 2-adrenoceptors.
@en
type
label
Studies on RX 781094: a select ...... nist of alpha 2-adrenoceptors.
@en
prefLabel
Studies on RX 781094: a select ...... nist of alpha 2-adrenoceptors.
@en
P2093
P2860
P1476
Studies on RX 781094: a select ...... nist of alpha 2-adrenoceptors.
@en
P2093
P2860
P304
P356
10.1111/J.1476-5381.1983.TB08809.X
P407
P577
1983-03-01T00:00:00Z