Exquisite selectivity for human toll-like receptor 8 in substituted furo[2,3-c]quinolines.
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Structure-Based Design of Novel Human Toll-like Receptor 8 AgonistsVirtual Screening Approaches towards the Discovery of Toll-Like Receptor ModulatorsIdentification of Adjuvantic Activity of Amphotericin B in a Novel, Multiplexed, Poly-TLR/NLR High-Throughput Screen.Enrichment assessment of multiple virtual screening strategies for Toll-like receptor 8 agonists based on a maximal unbiased benchmarking data set.Human Toll-like receptor 8-selective agonistic activities in 1-alkyl-1H-benzimidazol-2-aminesDeterminants of activity at human Toll-like receptors 7 and 8: quantitative structure-activity relationship (QSAR) of diverse heterocyclic scaffolds.The Imidazoquinoline Toll-Like Receptor-7/8 Agonist Hybrid-2 Potently Induces Cytokine Production by Human Newborn and Adult Leukocytes.Structure-Based Design of Human TLR8-Specific Agonists with Augmented Potency and Adjuvanticity.Directing the immune system with chemical compounds.Strategies for designing synthetic immune agonists.Synthesis of thieno[2,3-b]quinoline and selenopheno[2,3-b]quinoline derivatives via iodocyclization reaction and a DFT mechanistic study.Small-molecule inhibition of TLR8 through stabilization of its resting state.Recent advances in transition-metal-catalyzed reactions of alkynes with isoxazoles.Highly Convergent Synthesis of Intensively Blue Emissive Furo[2,3-c]isoquinolines by a Palladium-Catalyzed Cyclization Cascade of Unsaturated Ugi Products.Design and Synthesis of N1-Modified Imidazoquinoline Agonists for Selective Activation of Toll-like Receptors 7 and 8.Syntheses of Human TLR8-Specific Small-Molecule Agonists.
P2860
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P2860
Exquisite selectivity for human toll-like receptor 8 in substituted furo[2,3-c]quinolines.
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
2013年论文
@zh
2013年论文
@zh-cn
name
Exquisite selectivity for huma ...... tituted furo[2,3-c]quinolines.
@en
Exquisite selectivity for huma ...... tituted furo[2,3-c]quinolines.
@nl
type
label
Exquisite selectivity for huma ...... tituted furo[2,3-c]quinolines.
@en
Exquisite selectivity for huma ...... tituted furo[2,3-c]quinolines.
@nl
prefLabel
Exquisite selectivity for huma ...... tituted furo[2,3-c]quinolines.
@en
Exquisite selectivity for huma ...... tituted furo[2,3-c]quinolines.
@nl
P2093
P2860
P356
P1476
Exquisite selectivity for human toll-like receptor 8 in substituted furo[2,3-c]quinolines
@en
P2093
Alec R Hermanson
Anshuman Dixit
Hari Prasad Kokatla
Lauren M Fox
Rajalakshmi Balakrishna
Subbalakshmi S Malladi
Sunil A David
P2860
P304
P356
10.1021/JM400694D
P407
P577
2013-08-15T00:00:00Z