Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain.
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Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.Progress in HIV-1 Integrase Inhibitors: A Review of their Chemical Structure Diversity.Chelation Motifs Affecting Metal-dependent Viral Enzymes: N'-acylhydrazone Ligands as Dual Target Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H DomainNatural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding.Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and RDDP functions.Identification of spirocyclic or phosphate substituted quinolizine derivatives as novel HIV-1 integrase inhibitors: a patent evaluation of WO2016094197A1, WO2016094198A1 and WO2016154527A1.Inhibitory Effect of 2,3,5,6-Tetrafluoro-4-[4-(aryl)-1H-1,2,3-triazol-1-yl]benzenesulfonamide Derivatives on HIV Reverse Transcriptase Associated RNase H Activities.Prenylated phloroglucinols from Hypericum scruglii, an endemic species of Sardinia (Italy), as new dual HIV-1 inhibitors effective on HIV-1 replication.Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action.Uvaria angolensis as a promising source of inhibitors of HIV-1 RT-associated RNA-dependent DNA polymerase and RNase H functions.Improvement of the activity of the anti-HIV-1 integrase aptamer T30175 by introducing a modified thymidine into the loops.Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studiesFrom cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitorsRecent advances in the discovery of small-molecule inhibitors of HIV-1 integrase
P2860
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P2860
Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain.
description
2015 nî lūn-bûn
@nan
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
@zh
2015年论文
@zh-cn
name
Structure-activity relationshi ...... riptase ribonuclease H domain.
@en
Structure-activity relationshi ...... riptase ribonuclease H domain.
@nl
type
label
Structure-activity relationshi ...... riptase ribonuclease H domain.
@en
Structure-activity relationshi ...... riptase ribonuclease H domain.
@nl
prefLabel
Structure-activity relationshi ...... riptase ribonuclease H domain.
@en
Structure-activity relationshi ...... riptase ribonuclease H domain.
@nl
P2093
P50
P356
P1476
Structure-activity relationshi ...... riptase ribonuclease H domain.
@en
P2093
Antonella Messore
Christophe Marchand
Giovanni Pupo
Giuliana Cuzzucoli Crucitti
Luca Pescatori
Marta Cadeddu
Mathieu Métifiot
P304
P356
10.1021/JM501799K
P407
P50
P577
2015-02-11T00:00:00Z