Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
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Update on the Mechanism of Action of Aripiprazole: Translational Insights into Antipsychotic Strategies Beyond Dopamine Receptor AntagonismSnapin, a new regulator of receptor signaling, augments alpha1A-adrenoceptor-operated calcium influx through TRPC6Detection of receptor ligands by monitoring selective stabilization of a Renilla luciferase-tagged, constitutively active mutant, G-protein-coupled receptorSilodosin, a novel selective alpha 1A-adrenoceptor selective antagonist for the treatment of benign prostatic hyperplasia.alpha(1A)- and alpha(1B)-adrenergic receptors differentially modulate antidepressant-like behavior in the mouse.Feedback regulation of G protein-coupled receptor signaling by GRKs and arrestins.Alpha-1 adrenoceptor up-regulation induced by prazosin but not KMD-3213 or reserpine in rats.Novel role of mechanosensitive AT1B receptors in myogenic vasoconstriction.BIGL: Biochemically Intuitive Generalized Loewe null model for prediction of the expected combined effect compatible with partial agonism and antagonism.Effect of alpha-adrenoceptor subtype-selective inverse agonists on non-pregnant and late-pregnant cervical resistance in vitro in the rat.Evidence for altered brain reactivity to norepinephrine in Veterans with a history of traumatic stress.
P2860
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P2860
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
description
2000 nî lūn-bûn
@nan
2000年の論文
@ja
2000年学术文章
@wuu
2000年学术文章
@zh-cn
2000年学术文章
@zh-hans
2000年学术文章
@zh-my
2000年学术文章
@zh-sg
2000年學術文章
@yue
2000年學術文章
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2000年學術文章
@zh-hant
name
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@en
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@nl
type
label
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@en
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@nl
prefLabel
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@en
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@nl
P2093
P2860
P356
P1476
Inverse agonism and neutral antagonism at a constitutively active alpha-1a adrenoceptor.
@en
P2093
P2860
P304
P356
10.1038/SJ.BJP.0703584
P407
P577
2000-10-01T00:00:00Z