Stereoselective synthesis of peptidyl trifluoromethyl alcohols and ketones: inhibitory potency against human leucocyte elastase, cathepsin G, porcine pancreatic elastase and HIV-1 protease.

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Stereoselective synthesis of peptidyl trifluoromethyl alcohols and ketones: inhibitory potency against human leucocyte elastase, cathepsin G, porcine pancreatic elastase and HIV-1 protease.

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http://www.wikidata.org/entity/Q42540817

description

1998 nî lūn-bûn

@nan

1998年の論文

@ja

1998年論文

@yue

1998年論文

@zh-hant

1998年論文

@zh-hk

1998年論文

@zh-mo

1998年論文

@zh-tw

1998年论文

@wuu

1998年论文

@zh

1998年论文

@zh-cn

name

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@en

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@nl

type

Item

label

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@en

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@nl

prefLabel

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@en

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@nl

P1476

Stereoselective synthesis of p ...... c elastase and HIV-1 protease.

@en

P2093

Abouabdellah A

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Amour A

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Bonnet-Delpon D

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Bégue JP

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Le Gall M

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Reboud-Ravaux M

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de Rosny E

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P2860

Structure of chymotrypsin-trifluoromethyl ketone inhibitor complexes: comparison of slowly and rapidly equilibrating inhibitors

Structural analysis of the active site of porcine pancreatic elastase based on the X-ray crystal structures of complexes with trifluoroacetyl-dipeptide-anilide inhibitors

Chemical, biochemical, pharmacokinetic, and biological properties of L-680,833: a potent, orally active monocyclic beta-lactam inhibitor of human polymorphonuclear leukocyte elastase.

Human leukocyte and porcine pancreatic elastase: X-ray crystal structures, mechanism, substrate specificity, and mechanism-based inhibitors.

Human plasma proteinase inhibitors.

Synthetic inhibitors of elastase.

Fluoro ketone inhibitors of hydrolytic enzymes.

Pseudo-symmetrical difluoroketones. Highly potent and specific inhibitors of HIV-1 protease.

Synthesis of N-glyoxylyl peptides and their in vitro evaluation as HIV-1 protease inhibitors.

Mechanism of slow-binding inhibition of human leukocyte elastase by trifluoromethyl ketones.

P304

593-600

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P31

scholarly article

P356

10.1111/J.2042-7158.1998.TB06892.X

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P433

http://www.w3.org/2001/XMLSchema#string

P478

http://www.w3.org/2001/XMLSchema#string

P577

1998-06-01T00:00:00Z

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P698

9680068

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P921

stereoselectivity