Superpotent [Dmt¹] dermorphin tetrapeptides containing the 4-aminotetrahydro-2-benzazepin-3-one scaffold with mixed μ/δ opioid receptor agonistic properties.
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One-pot isomerization-cross metathesis-reduction (ICMR) synthesis of lipophilic tetrapeptidesBifunctional Peptide-Based Opioid Agonist-Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic PainIn vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist-neurokinin 1 receptor antagonist chimeraVariation of the net charge, lipophilicity, and side chain flexibility in Dmt(1)-DALDA: Effect on Opioid Activity and Biodistribution.χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.A one-pot multicomponent approach to a new series of morphine derivatives and their biological evaluation.Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings.
P2860
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P2860
Superpotent [Dmt¹] dermorphin tetrapeptides containing the 4-aminotetrahydro-2-benzazepin-3-one scaffold with mixed μ/δ opioid receptor agonistic properties.
description
2011 nî lūn-bûn
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2011年の論文
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2011年学术文章
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2011年学术文章
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name
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties.
@en
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties.
@nl
type
label
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties.
@en
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties.
@nl
prefLabel
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties.
@en
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties.
@nl
P2093
P356
P1476
Superpotent [Dmt¹] dermorphin ...... receptor agonistic properties
@en
P2093
Alexandra Gramowski-Voss
Andrzej Lipkowski
Bart Vandormael
Danai-Dionysia Fourla
Dirk Tourwé
Olaf H-U Schröder
Zafiroula Georgoussi
P304
P356
10.1021/JM200894E
P407
P577
2011-10-20T00:00:00Z