The Bruton Tyrosine Kinase (BTK) Inhibitor Acalabrutinib Demonstrates Potent On-Target Effects and Efficacy in Two Mouse Models of Chronic Lymphocytic Leukemia.
about
New drug discovery approaches targeting recurrent mutations in chronic lymphocytic leukemia.Pharmacotherapy of relapsed/refractory chronic lymphocytic leukemia.Mechanisms of Resistance to Targeted Therapies in Chronic Lymphocytic Leukemia.The specific Bruton tyrosine kinase inhibitor acalabrutinib (ACP-196) shows favorable in vitro activity against chronic lymphocytic leukemia B cells with CD20 antibodiesCombined BTK and PI3Kδ Inhibition with Acalabrutinib and ACP-319 Improves Survival and Tumor Control in CLL Mouse Model.Novel synthetic drugs currently in clinical development for chronic lymphocytic leukemia.Role of Bruton's tyrosine kinase in B cells and malignancies.Acalabrutinib: First Global Approval.Potent anti-leukemic activity of a specific cyclin-dependent kinase 9 inhibitor in mouse models of chronic lymphocytic leukemia.
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P2860
The Bruton Tyrosine Kinase (BTK) Inhibitor Acalabrutinib Demonstrates Potent On-Target Effects and Efficacy in Two Mouse Models of Chronic Lymphocytic Leukemia.
description
2016 nî lūn-bûn
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2016年の論文
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2016年学术文章
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2016年学术文章
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2016年学术文章
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2016年学术文章
@zh-hans
2016年学术文章
@zh-my
2016年学术文章
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2016年學術文章
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2016年學術文章
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name
The Bruton Tyrosine Kinase (BT ...... Chronic Lymphocytic Leukemia.
@en
The Bruton Tyrosine Kinase
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type
label
The Bruton Tyrosine Kinase (BT ...... Chronic Lymphocytic Leukemia.
@en
The Bruton Tyrosine Kinase
@nl
prefLabel
The Bruton Tyrosine Kinase (BT ...... Chronic Lymphocytic Leukemia.
@en
The Bruton Tyrosine Kinase
@nl
P2093
P2860
P50
P1476
The Bruton Tyrosine Kinase (BT ...... Chronic Lymphocytic Leukemia.
@en
P2093
Adrian Wiestner
Allard Kaptein
Amy J Johnson
Arnau Montraveta
Brian J Lannutti
Fabienne McClanahan
Fanny Krantz
Helena Mora-Jensen
Jennifer A Woyach
Lisa L Smith
P2860
P304
P356
10.1158/1078-0432.CCR-16-0463
P407
P577
2016-11-30T00:00:00Z