Species differences in affinities of non-peptide antagonists for substance P receptors.
about
Tachykinin receptors and tachykinin receptor antagonistsAnxiolytic-like effects of the neurokinin 1 receptor antagonist GR-205171 in the elevated plus maze and contextual fear-potentiated startle model of anxiety in gerbils.Innervation of the synoviumNew insights into the antidepressant actions of substance P (NK1 receptor) antagonists.Behavioral and pharmacological validation of the gerbil forced-swim test: effects of neurokinin-1 receptor antagonists.Effects of RP 67580, a tachykinin NK1 receptor antagonist, on a primary afferent-evoked response of ventral roots in the neonatal rat spinal cord.The interaction of escitalopram and R-citalopram at the human serotonin transporter investigated in the mouse.Role of substance P in inflammatory arthritis.Non-peptide antagonists, CP-96,345 and RP 67580, distinguish species variants in tachykinin NK1 receptors.(+/-)-CP-96,345, a selective tachykinin NK1 receptor antagonist, has non-specific actions on neurotransmission.Tachykinin receptors in rabbit airways--characterization by functional, autoradiographic and binding studies.Antinociceptive activity of the tachykinin NK1 receptor antagonist, CP-99,994, in conscious gerbils.Relationships between neurokinin receptor-expressing interstitial cells of Cajal and tachykininergic nerves in the gut.Effects of interactions of naturally-occurring neuropeptides on blood flow in the rat knee joint.Neurokinin receptors. Comparison of data from classical pharmacology, binding, and molecular biology.Pharmacological properties of a potent and selective nonpeptide substance P antagonist.Tachykinin receptors: a radioligand binding perspective.Substance P-evoked calcium mobilization and ionic current activation in the human astrocytoma cell line U 373 MG: pharmacological characterization.Characterization of a human NK1 tachykinin receptor in the astrocytoma cell line U 373 MG.Antinociceptive activity of NK1 receptor antagonists: non-specific effects of racemic RP67580.Effect of the tachykinin NK1 receptor antagonists, RP 67580 and SR 140333, on electrically-evoked substance P release from rat spinal cord.Inhibition of Ca(2+)-sensitive K+ currents in NG 108-15 cells by substance P and related tachykininsComparative behavioural profile of centrally administered tachykinin NK1, NK2 and NK3 receptor agonists in the guinea-pig.Higher potency of RP 67580, in the mouse and the rat compared with other nonpeptide and peptide tachykinin NK1 antagonists.Tachykinin NK1 receptor in the guinea-pig isolated proximal urethra: characterization by receptor selective agonists and antagonists.The interaction of the NK1 receptor antagonist CP-96,345 with L-type calcium channels and its functional consequences.A pharmacological study of NK1 and NK2 tachykinin receptor characteristics in the rat isolated urinary bladder.FR 113680: a novel tripeptide substance P antagonist with NK1 receptor selectivity.Presence of NK3-sensitive neurones in different proportions in the medial habenula of guinea-pig, rat and gerbil.Comparison of tachykinin NK1 and NK2 receptors in the circular muscle of the guinea-pig ileum and proximal colon.The non-peptide NK1 receptor antagonist, (+/-)-CP-96,345, produces antinociceptive and anti-oedema effects in the rat.Tachykinin NK1 receptor subtypes in the rat urinary bladder.The pharmacology of GR203040, a novel, potent and selective non-peptide tachykinin NK1 receptor antagonist.Investigation into species variants in tachykinin NK1 receptors by use of the non-peptide antagonist, CP-96,345.Pharmacological profile of a high affinity dipeptide NK1 receptor antagonist, FK888Use of selective antagonists to dissociate the central cardiovascular and behavioural effects of tachykinins on NK1 and NK2 receptors in the rat.Prejunctional control of pH 6-induced bronchoconstriction by NK1, NK2, mu-opioid, alpha2-adrenoceptor and glucocorticoid receptors in guinea-pig isolated perfused lung.beta-Amyloid (25-35) or substance P stimulates [3H]MK-801 binding to rat cortical membranes in the presence of glutamate and glycine.
P2860
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P2860
Species differences in affinities of non-peptide antagonists for substance P receptors.
description
1991 nî lūn-bûn
@nan
1991年の論文
@ja
1991年学术文章
@wuu
1991年学术文章
@zh
1991年学术文章
@zh-cn
1991年学术文章
@zh-hans
1991年学术文章
@zh-my
1991年学术文章
@zh-sg
1991年學術文章
@yue
1991年學術文章
@zh-hant
name
Species differences in affinities of non-peptide antagonists for substance P receptors.
@en
Species differences in affinities of non-peptide antagonists for substance P receptors.
@nl
type
label
Species differences in affinities of non-peptide antagonists for substance P receptors.
@en
Species differences in affinities of non-peptide antagonists for substance P receptors.
@nl
prefLabel
Species differences in affinities of non-peptide antagonists for substance P receptors.
@en
Species differences in affinities of non-peptide antagonists for substance P receptors.
@nl
P2093
P1476
Species differences in affinities of non-peptide antagonists for substance P receptors.
@en
P2093
P304
P356
10.1016/0014-2999(91)90532-U
P407
P577
1991-05-01T00:00:00Z