Dopamine receptor parameters detected by [3H]spiperone depend on tissue concentration: analysis and examples.
about
History of the discovery of the antipsychotic dopamine D2 receptor: a basis for the dopamine hypothesis of schizophreniaSchizophrenia, amphetamine-induced sensitized state and acute amphetamine exposure all show a common alteration: increased dopamine D2 receptor dimerizationDopamine receptor contribution to the action of PCP, LSD and ketamine psychotomimeticsAll Roads to Schizophrenia Lead to Dopamine Supersensitivity and Elevated Dopamine D2High ReceptorsNMDA receptor antagonists ketamine and PCP have direct effects on the dopamine D(2) and serotonin 5-HT(2)receptors-implications for models of schizophrenia.Cocaine self-administration produces a persistent increase in dopamine D2 High receptors.Dopamine receptors in human lymphocytes: radioligand binding and quantitative RT-PCR assays.How membrane partitioning modulates receptor activation: parallel versus serial effects of hydrophobic ligands.Clozapine, a fast-off-D2 antipsychotic.Tactics for preclinical validation of receptor-binding radiotracers.The Trace Amine 1 receptor knockout mouse: an animal model with relevance to schizophrenia.Comparison of the in-vitro receptor selectivity of substituted benzamide drugs for brain neurotransmitter receptors.N1-methyl-2-125I-lysergic acid diethylamide, a preferred ligand for in vitro and in vivo characterization of serotonin receptors.Cannabidiol is a partial agonist at dopamine D2High receptors, predicting its antipsychotic clinical doseIn vivo receptor assay with multiple ligand concentrations: an equilibrium approach.Amphetamine-sensitized animals show a marked increase in dopamine D2 high receptors occupied by endogenous dopamine, even in the absence of acute challenges.Pitfalls in membrane binding sites studies in post-mortem human brain.Acute social defeat does not alter cerebral 5-HT2A receptor binding in male Wistar rats.Comparison of neuroleptic binding characteristics in rat striatum and renal cortex.Neurotransmitters, receptors and neuropeptides in post-mortem brains of chronic schizophrenic patients.
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P2860
Dopamine receptor parameters detected by [3H]spiperone depend on tissue concentration: analysis and examples.
description
1984 nî lūn-bûn
@nan
1984年の論文
@ja
1984年学术文章
@wuu
1984年学术文章
@zh
1984年学术文章
@zh-cn
1984年学术文章
@zh-hans
1984年学术文章
@zh-my
1984年学术文章
@zh-sg
1984年學術文章
@yue
1984年學術文章
@zh-hant
name
Dopamine receptor parameters d ...... ration: analysis and examples.
@en
Dopamine receptor parameters d ...... ration: analysis and examples.
@nl
type
label
Dopamine receptor parameters d ...... ration: analysis and examples.
@en
Dopamine receptor parameters d ...... ration: analysis and examples.
@nl
prefLabel
Dopamine receptor parameters d ...... ration: analysis and examples.
@en
Dopamine receptor parameters d ...... ration: analysis and examples.
@nl
P2093
P2860
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Dopamine receptor parameters d ...... ration: analysis and examples.
@en
P2093
P2860
P304
P356
10.1111/J.1471-4159.1984.TB06700.X
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P577
1984-07-01T00:00:00Z