Synthesis of stereodefined piperidines from aziridines and their transformation into conformationally constrained amino acids, amino alcohols and 2,7-diazabicyclo[3.3.1]nonanes.
about
Regioselectivity in the ring opening of non-activated aziridines.Radical-mediated nitrile translocation as the key step in the stereoselective transformation of 2-(4-chloro-2-cyanobutyl)aziridines to methyl cis-(1-arylmethyl-4-phenylpiperidin-2-yl)acetates.Straightforward synthesis of 1-alkyl-2-(trifluoromethyl)aziridines starting from 1,1,1-trifluoroacetone.Synthesis of new functionalized aziridine-2- and azetidine-3-carboxylic acid derivatives of potential interest for biological and foldameric applications.LiAlH4 -Induced Selective Ring Rearrangement of 2-(2-Cyanoethyl)aziridines toward 2-(Aminomethyl)pyrrolidines and 3-Aminopiperidines as Eligible Heterocyclic Building Blocks.Selective synthesis of functionalized trifluoromethylated pyrrolidines, piperidines, and azepanes starting from 1-tosyl-2-(trifluoromethyl)aziridine.Synthesis of 2-aryl-3-(2-cyanoethyl)aziridines and their chemical and enzymatic hydrolysis towards γ-lactams and γ-lactones.One-pot multiple reactions: asymmetric synthesis of 2,6-cis-disubstituted piperidine alkaloids from chiral aziridine.Structure and pharmacological studies of the anaesthetic 1-(3-n-butoxypropyl)-4-benzoyloxypiperidin hydrochloride and its complex with β-cyclodextrin in solution. NMR and IR-spectroscopy data
P2860
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P2860
Synthesis of stereodefined piperidines from aziridines and their transformation into conformationally constrained amino acids, amino alcohols and 2,7-diazabicyclo[3.3.1]nonanes.
description
2010 nî lūn-bûn
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2010年の論文
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2010年学术文章
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2010年学术文章
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2010年学术文章
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2010年学术文章
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2010年学术文章
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2010年学术文章
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name
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@en
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@nl
type
label
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@en
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@nl
prefLabel
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@en
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@nl
P2093
P356
P1476
Synthesis of stereodefined pip ...... ,7-diazabicyclo[3.3.1]nonanes.
@en
P2093
Karel Vervisch
Karl W Törnroos
Matthias D'hooghe
P304
P356
10.1021/JO101646U
P407
P577
2010-10-26T00:00:00Z