about
α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome.Revisiting Previously Investigated Plants: A Molecular Networking-Based Study of Geissospermum laeve.Design, synthesis and anticancer properties of IsoCombretaQuinolines as potent tubulin assembly inhibitors.Discovery of azaisoerianin derivatives as potential antitumors agents.Synthesis, biological evaluation, and structure-activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors.Interaction of chemokine receptor CXCR4 in monomeric and dimeric state with its endogenous ligand CXCL12: coarse-grained simulations identify differences.Comparative study of structural models of Leishmania donovani and human GDP-mannose pyrophosphorylases.Characterization of the Annonaceous acetogenin, annonacinone, a natural product inhibitor of plasminogen activator inhibitor-1.A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime.Enantioselective Three-Component Amination of Enecarbamates Enables the Synthesis of Structurally Complex Small Molecules.A fluorine scan of a tubulin polymerization inhibitor isocombretastatin A-4: Design, synthesis, molecular modelling, and biological evaluation.Enantioselective Brønsted Acid Catalysis as a Tool for the Synthesis of Natural Products and Pharmaceuticals.Diversity-oriented synthesis of fused thioglycosyl benzo[e][1,4]oxathiepin-5-ones and benzo[f][1,4]thiazepin-5(2H)-ones by a sequence of palladium-catalyzed glycosyl thiol arylation and deprotection-lactonization reactions.A unified bioinspired "aplysinopsin cascade": total synthesis of (±)-tubastrindole B and related biosynthetic congeners.Unified biomimetic assembly of voacalgine A and bipleiophylline via divergent oxidative couplings.Design, Synthesis, and Biological Activity of New N-(Phenylmethyl)-benzoxazol-2-thiones as Macrophage Migration Inhibitory Factor (MIF) Antagonists: Efficacies in Experimental Pulmonary Hypertension.IsoCombretaQuinazolines: Potent Cytotoxic Agents with Antitubulin Activity.Theionbrunonines A and B: Dimeric Vobasine Alkaloids Tethered by a Thioether Bridge from Mostuea brunonisSynthesis and conformational studies of a stable peptidomimetic β-hairpin based on a bifunctional diketopiperazine turn inducerDP4-Assisted Structure Elucidation of Isodemethylchodatin, a New Norlichexanthone Derivative Meager in H-Atoms, from the LichenCarbonylhydrazide-based molecular tongs inhibit wild-type and mutated HIV-1 protease dimerizationCarbonic anhydrase binding site parameterization in OPLS-AA force fieldRegio-, Diastereo-, and Enantioselective Nitroso-Diels-Alder Reaction of 1,3-Diene-1-carbamates Catalyzed by Chiral Phosphoric AcidsSpontaneous biomimetic formation of (±)-dictazole B under irradiation with artificial sunlightN-Difluoromethyl-triazole as a constrained scaffold in peptidomimeticsNervisides I-J: Unconventional Side-Chain-Bearing Cycloartane Glycosides from Nervilia concolorSynthesis of 3,5-Disubstituted 1,2-Dioxolanes through the Use of Acetoxy PeroxyacetalsDifferential activity and selectivity of N-terminal modified CXCL12 chemokines at the CXCR4 and ACKR3 receptorsThermodynamic epimeric equilibration and crystallisation-induced dynamic resolution of lobelanine, norlobelanine and related analogues
P50
Q35031028-87BC538A-EF30-4721-9A4E-CF25ED3CF8E9Q36304066-15C0B25C-7ACF-4BED-A303-25C6CB22D09EQ38717671-04323E38-F47B-4478-B6BB-BFF32E141C17Q39010208-17460688-7DB5-47FE-8EFF-45BC58D7311DQ39263355-6BC2318E-25C3-4512-A91E-C0F61DE49E33Q40058610-171EE827-1AD4-4742-90BE-CA53ABDD07BFQ40327849-C55C5C40-265B-468B-B037-96AA3A0BF7CBQ42364420-3B0F479A-6FDF-4202-A543-D2A848725864Q42782433-30AC8DE2-C8FC-4063-8848-E4E773A7831AQ46432059-297F3596-C22C-4031-B3A7-4001055B9324Q47333989-0BEA5747-DA3B-4554-A026-2F3B929F5927Q48238623-B0675B32-F0AD-4188-A2D3-FB8F7E626B15Q50935791-11B13419-6725-4F6A-9AED-E7EC296EFD9EQ51409290-5432A422-965C-4703-840E-49A4668337B5Q52560498-4185AF70-ED94-4854-8623-1F12EDABBAF9Q52662257-47988A2E-2D35-45F3-8F72-EEFEBA60099BQ52936807-8D416CE3-5FDE-469B-A6AE-5367B831974EQ57285820-A38AB2B6-A771-4AF4-B295-3649F4F0E25DQ58037802-C38190F1-3876-44F4-A5FC-39D4A9E4CF13Q64252387-1B2184B9-9A7B-4B40-A5F4-8ED627062F41Q84576828-0EF43F06-2975-458A-8CCC-87E700A54B47Q85534192-5FEC3DAF-9D22-4CA8-9438-D9241FCC8F86Q86102692-C76F1696-E2C5-4DBD-8307-5A50B917EBADQ87853644-14591A72-8591-4877-90E2-312C5F2C4BB7Q87880175-AA2DCE0B-30F6-4D53-B658-93DD597813C7Q91994059-4B918CCD-416B-48AE-A269-288C9A65ADFDQ92656497-BB139CC0-B5D2-4AAB-B166-2DA9CC124AF2Q94566787-324C0CF9-1A68-484C-AC41-1A24EBF35557Q95615454-D2B53288-84F2-42B0-BADC-A482DA8B019B
P50
description
researcher
@en
wetenschapper
@nl
հետազոտող
@hy
name
Guillaume Bernadat
@ast
Guillaume Bernadat
@en
Guillaume Bernadat
@es
Guillaume Bernadat
@nl
type
label
Guillaume Bernadat
@ast
Guillaume Bernadat
@en
Guillaume Bernadat
@es
Guillaume Bernadat
@nl
prefLabel
Guillaume Bernadat
@ast
Guillaume Bernadat
@en
Guillaume Bernadat
@es
Guillaume Bernadat
@nl
P106
P31
P496
0000-0001-8955-0364