about
Dioxo-triazines as a novel series of cathepsin K inhibitorsStructure based evolution of a novel series of positive modulators of the AMPA receptorFunctional analysis of a novel positive allosteric modulator of AMPA receptors derived from a structure-based drug design strategyThe Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS HitsStructurally Diverse Mitochondrial Branched Chain Aminotransferase (BCATm) Leads with Varying Binding Modes Identified by Fragment ScreeningEvolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory DiseaseScope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulationRational Design of a Novel AMPA Receptor Modulator through a Hybridization Approach.Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators.Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA2 Inhibitor.Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode.Surface Functionalization with Carboxylic Acids by Photochemical Microcontact Printing and Tetrazole Chemistry.Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.One-Pot, Three-Step Synthesis of Cyclopropylboronic Acid Pinacol Esters from Synthetically Tractable Propargylic Silyl Ethers.Synthesis of the originally proposed structures of elatenyne and an enyne from Laurencia majusculaOrganobase-Catalyzed Amidation of Esters with Amino AlcoholsAmidation of esters with amino alcohols using organobase catalysisCatalytic amidation of unactivated ester derivatives mediated by trifluoroethanolAmidation of unactivated ester derivatives mediated by trifluoroethanolCyrene as a bio-based solvent for HATU mediated amide couplingAtom Efficient Synthesis of Selectively Difluorinated Carbocycles through a Gold(I)-Catalyzed CyclizationA Multicomponent Route to Functionalized Amides and OxazolidinonesMetal-free C-C bond formation via coupling of nitrile imines and boronic acidsPhotocatalytic E → Z Isomerization of β-Ionyl DerivativesA fragment-like approach to PYCR1 inhibition
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description
researcher, ORCID id # 0000-0002-6567-8272
@en
wetenschapper
@nl
name
Craig Jamieson
@ast
Craig Jamieson
@en
Craig Jamieson
@es
Craig Jamieson
@nl
type
label
Craig Jamieson
@ast
Craig Jamieson
@en
Craig Jamieson
@es
Craig Jamieson
@nl
prefLabel
Craig Jamieson
@ast
Craig Jamieson
@en
Craig Jamieson
@es
Craig Jamieson
@nl
P106
P1153
57188805955
7006413261
P31
P496
0000-0002-6567-8272