about
Betraying the parasite's redox system: diaryl sulfide-based inhibitors of trypanothione reductase: subversive substrates and antitrypanosomal properties.Antibody-drug conjugates: linking cytotoxic payloads to monoclonal antibodies.Synthesis, inhibition potency, binding mode, and antiprotozoal activities of fluorescent inhibitors of trypanothione reductase based on mepacrine-conjugated diaryl sulfide scaffolds.Pentafluorosulfanyl as a novel building block for enzyme inhibitors: trypanothione reductase inhibition and antiprotozoal activities of diarylamines.Diaryl sulfide-based inhibitors of trypanothione reductase: inhibition potency, revised binding mode and antiprotozoal activities.Structure-based design, synthesis, and in vitro evaluation of nonpeptidic neprilysin inhibitors
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description
researcher ORCID ID = 0000-0003-3670-8038
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wetenschapper
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name
Bernhard Stump
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Bernhard Stump
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Bernhard Stump
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Bernhard Stump
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type
label
Bernhard Stump
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Bernhard Stump
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Bernhard Stump
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Bernhard Stump
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prefLabel
Bernhard Stump
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Bernhard Stump
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Bernhard Stump
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Bernhard Stump
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0000-0003-3670-8038