about
First insight into structure-activity relationships of selective meprin β inhibitors.Natural Products from Microalgae with Potential against Alzheimer's Disease: Sulfolipids Are Potent Glutaminyl Cyclase Inhibitors.Inhibition of glutaminyl cyclase prevents pGlu-Abeta formation after intracortical/hippocampal microinjection in vivo/in situ.Isolation, catalytic properties, and competitive inhibitors of the zinc-dependent murine glutaminyl cyclase.The first potent inhibitors for human glutaminyl cyclase: synthesis and structure-activity relationship.3-Hydroxy-N'-arylidenepropanehydrazonamides with Halo-Substituted Phenanthrene Scaffolds Cure P. berghei Infected Mice When Administered Perorally.Inhibitors for human glutaminyl cyclase by structure based design and bioisosteric replacement.Structure-activity relationships of benzimidazole-based glutaminyl cyclase inhibitors featuring a heteroaryl scaffold.Semi-empirical derived descriptors for the modelling of properties of N-containing heterocycles.Structure-guided design, synthesis and characterization of next-generation meprin β inhibitors.Dipeptidyl-Peptidase Activity of Meprin β Links N-truncation of Aβ with Glutaminyl Cyclase-Catalyzed pGlu-Aβ FormationExpression of human and Porphyromonas gingivalis glutaminyl cyclases in periodontitis and rheumatoid arthritis-A pilot studyTertiary-Amine-Based Inhibitors of the Astacin Protease Meprin αHydrazides are potent transition-state analogs for glutaminyl cyclase implicated in the pathogenesis of Alzheimer's Disease
P50
Q30313253-494FAE20-767C-4D69-AD6F-9B94A21EDAB4Q30313757-433971AB-96F7-461F-B858-61E2D664057BQ30319495-02005A54-09BB-4BBC-82A3-AC69B6E35D3CQ30320146-AA34D3E8-7FF9-4ED1-9A76-0162DE64583BQ33231898-FF0250A6-BA1D-49E5-B943-A29A8F448FFFQ39172819-BFC3BCC7-4215-4A0F-9949-BDBCC3358E57Q39782565-5C72A84A-45D4-4DDE-957D-788B91F89AC8Q45275098-2CCCBA92-E162-4FE7-8795-B82044A71E84Q45752203-3382F001-9E77-4C94-BE04-6550E2AD1A60Q52563984-4ABC78DE-A9FB-4845-9A6D-B64580C99A0FQ57489797-5518B724-AA72-446F-A2F6-FC2E708DDC8EQ58600305-896480BE-761B-4E48-898F-CB7A5FDFF524Q59388051-CB9C9582-EA71-402D-A240-8AC4C3A77AB4Q96580271-DC0C7DF9-F2C9-4474-B6E0-820B3446FD15
P50
description
onderzoeker
@nl
researcher ORCID ID = 0000-0002-2629-4153
@en
name
Mirko Buchholz
@ast
Mirko Buchholz
@en
Mirko Buchholz
@es
Mirko Buchholz
@nl
type
label
Mirko Buchholz
@ast
Mirko Buchholz
@en
Mirko Buchholz
@es
Mirko Buchholz
@nl
prefLabel
Mirko Buchholz
@ast
Mirko Buchholz
@en
Mirko Buchholz
@es
Mirko Buchholz
@nl
P106
P31
P496
0000-0002-2629-4153