about
Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulationChemoselective oxidation of aryl organoboron systems enabled by boronic acid-selective phase transferRational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators.Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.Chemoselective boronic ester synthesis by controlled speciation.Synthesis of functionalised 4H-quinolizin-4-ones via tandem Horner-Wadsworth-Emmons olefination/cyclisation.Soft scorpionate anions as platforms for novel heterocycles.In situ generation of Mes2Mg as a non-nucleophilic carbon-centred base reagent for the efficient one-pot conversion of ketones to silyl enol ethers.Interrogating Pd(II) Anion Metathesis Using a Bifunctional Chemical Probe: A Transmetalation Switch.Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode.Chemoselective Suzuki-Miyaura Cross-Coupling via Kinetic Transmetallation.Spectroscopic Studies of the Chan-Lam Amination: A Mechanism-Inspired Solution to Boronic Ester Reactivity.Strategy for Conditional Orthogonal Sequential CuAAC Reactions Using a Protected Aromatic Ynamine.Determining the Origin of Rate-Independent Chemoselectivity in CuAAC Reactions: An Alkyne-Specific Shift in Rate-Determining Step.Contra-Thermodynamic, Photocatalytic E→Z Isomerization of Styrenyl Boron Species: Vectors to Facilitate Exploration of 2D Chemical Space.Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.Correction to "Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides".Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides.Tandem Chemoselective Suzuki-Miyaura Cross-Coupling Enabled by Nucleophile Speciation Control.Chemoselective One-Pot Synthesis of Functionalized Amino-azaheterocycles Enabled by COware.Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second Bromodomain.Scalable total synthesis and comprehensive structure-activity relationship studies of the phytotoxin coronatine.A flow platform for degradation-free CuAAC bioconjugationBiocatalytic Synthesis of Chiral N-Functionalized Amino AcidsBismesitylmagnesium: a thermally stable and non-nucleophilic carbon-centred base reagent for the efficient preparation of silyl enol ethersTowards energetically viable asymmetric deprotonations: selectivity at more elevated temperatures with C2-symmetric magnesium bisamidesAmidation of esters with amino alcohols using organobase catalysisA modular synthesis of functionalised phenols enabled by controlled boron speciationOne-Pot Homologation of Boronic Acids: A Platform for Diversity-Oriented SynthesisSpeciation control during Suzuki-Miyaura cross-coupling of haloaryl and haloalkenyl MIDA boronic estersSynthesis of 2-BMIDA 6,5-bicyclic heterocycles by Cu(i)/Pd(0)/Cu(ii) cascade catalysis of 2-iodoaniline/phenolsAmidation of unactivated ester derivatives mediated by trifluoroethanolCyrene as a bio-based solvent for HATU mediated amide couplingA one-pot tandem chemoselective allylation/cross-coupling via temperature control of a multi-nucleophile/electrophile systemChan-Evans-Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine ProblemCatalytic Enantioselective Synthesis of α-Chiral Azaheteroaryl Ethylamines by Asymmetric ProtonationA Multicomponent Route to Functionalized Amides and OxazolidinonesDeoxyfluorination with CuF2 : Enabled by Using a Lewis Base Activating GroupN-Alkyl-α-amino acids in Nature and their biocatalytic preparationMechanistic Development and Recent Applications of the Chan-Lam Amination
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P50
description
investigador
@es
researcher
@en
wetenschapper
@nl
name
Allan J B Watson
@en
Allan J B Watson
@nl
type
label
Allan J B Watson
@en
Allan J B Watson
@nl
prefLabel
Allan J B Watson
@en
Allan J B Watson
@nl
P108
P31
P496
0000-0002-1582-4286