about
Design and Development of Highly Potent HIV-1 Protease Inhibitors with a Crown-Like Oxotricyclic Core as the P2-Ligand To Combat Multidrug-Resistant HIV Variants.Design, Synthesis, Biological Evaluation, and X-ray Studies of HIV-1 Protease Inhibitors with Modified P2' Ligands of Darunavir.Design of Highly Potent, Dual Acting and Central Nervous System Penetrating HIV-1 Protease Inhibitors with Excellent Potency against Multidrug-Resistant HIV-1 Variants.Enantioselective Synthesis of Spliceostatin G and Evaluation of Bioactivity of Spliceostatin G and Its Methyl Ester.Design and Synthesis of Highly Potent HIV-1 Protease Inhibitors Containing Tricyclic Fused Ring Systems as Novel P2 Ligands: Structure-Activity Studies, Biological and X-ray Structural Analysis.Design and Synthesis of Potent HIV-1 Protease Inhibitors Containing Bicyclic Oxazolidinone Scaffold as the P2 Ligands: Structure-Activity Studies and Biological and X-ray Structural StudiesEnantioselective Synthesis of a Cyclopropane Derivative of Spliceostatin A and Evaluation of BioactivityThe Curtius rearrangement: mechanistic insight and recent applications in natural product synthesesEnantioselective Synthesis of Thailanstatin A Methyl Ester and Evaluation of in Vitro Splicing InhibitionDifferentiating Isomeric Deprotonated Glucuronide Drug Metabolites via Ion/Molecule Reactions in Tandem Mass SpectrometryPotent HIV-1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein-Ligand X-ray Structural StudiesDevelopment of an Efficient Enzyme Production and Structure-Based Discovery Platform for BACE1 InhibitorsFluorescent Probes for Monitoring Serine UbiquitinationHighly Selective and Potent Human β-Secretase 2 (BACE2) Inhibitors against Type 2 Diabetes: Design, Synthesis, X-ray Structure and Structure-Activity Relationship StudiesThe Curtius Rearrangement: Applications in Modern Drug Discovery and Medicinal ChemistryEnantioselective Total Synthesis of (+)-Monocerin, a Dihydroisocoumarin Derivative with Potent Antimalarial PropertiesUrea Derivatives in Modern Drug Discovery and Medicinal ChemistryA Photochemical Route to Optically Active Hexahydro-4H-furopyranol, a High-Affinity P2 Ligand for HIV-1 Protease InhibitorsEnantioselective Total Syntheses of (+)-Fendleridine and (+)-AcetylaspidoalbidineStructure-Based Design of Highly Potent HIV-1 Protease Inhibitors Containing New Tricyclic Ring P2-Ligands: Design, Synthesis, Biological, and X-ray Structural StudiesCopper-Catalyzed Stille Cross-Coupling Reaction and Application in the Synthesis of the Spliceostatin Core Structure
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P50
description
researcher
@en
wetenschapper
@nl
name
Arun K Ghosh
@en
Arun K Ghosh
@nl
type
label
Arun K Ghosh
@en
Arun K Ghosh
@nl
prefLabel
Arun K Ghosh
@en
Arun K Ghosh
@nl
P31
P496
0000-0003-2472-1841