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Q36739519-9629F801-D484-46E3-B6B6-EB066E184927
Q36739519-9629F801-D484-46E3-B6B6-EB066E184927
BestRank
Statement
http://www.wikidata.org/entity/statement/Q36739519-9629F801-D484-46E3-B6B6-EB066E184927
Structure-based design of N-substituted 1-hydroxy-4-sulfamoyl-2-naphthoates as selective inhibitors of the Mcl-1 oncoprotein.
P2860
Q36739519-9629F801-D484-46E3-B6B6-EB066E184927
BestRank
Statement
http://www.wikidata.org/entity/statement/Q36739519-9629F801-D484-46E3-B6B6-EB066E184927
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type
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wasDerivedFrom
99eb4192585e5bec7ce7111a0c5d153e3c71959d
P2860
Potent and selective small-molecule MCL-1 inhibitors demonstrate on-target cancer cell killing activity as single agents and in combination with ABT-263 (navitoclax).