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Q41848109-77493E5C-B612-4075-8D16-952259A8DDDC
Q41848109-77493E5C-B612-4075-8D16-952259A8DDDC
BestRank
Statement
http://www.wikidata.org/entity/statement/Q41848109-77493E5C-B612-4075-8D16-952259A8DDDC
A first-in-class NAE inhibitor, MLN4924, blocks lentiviral infection in myeloid cells by disrupting neddylation-dependent Vpx-mediated SAMHD1 degradation.
P2860
Q41848109-77493E5C-B612-4075-8D16-952259A8DDDC
BestRank
Statement
http://www.wikidata.org/entity/statement/Q41848109-77493E5C-B612-4075-8D16-952259A8DDDC
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type
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wasDerivedFrom
d45a5e49325f6e0463827a49beac5156b9d6836b
P2860
A dominant-negative UBC12 mutant sequesters NEDD8 and inhibits NEDD8 conjugation in vivo