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Q41934777-67351D90-359C-40C6-852D-13E90120A814
Q41934777-67351D90-359C-40C6-852D-13E90120A814
BestRank
Statement
http://www.wikidata.org/entity/statement/Q41934777-67351D90-359C-40C6-852D-13E90120A814
Metabolic activation of mifepristone [RU486; 17beta-hydroxy-11beta-(4-dimethylaminophenyl)-17alpha-(1-propynyl)-estra-4,9-dien-3-one] by mammalian cytochromes P450 and the mechanism-based inactivation of human CYP2B6.
P2860
Q41934777-67351D90-359C-40C6-852D-13E90120A814
BestRank
Statement
http://www.wikidata.org/entity/statement/Q41934777-67351D90-359C-40C6-852D-13E90120A814
rank
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type
BestRank
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wasDerivedFrom
6524a8c96b0d6a2e06088e45b48be90616272c38
P2860
The cytochrome P450 2B6 (CYP2B6) is the main catalyst of efavirenz primary and secondary metabolism: implication for HIV/AIDS therapy and utility of efavirenz as a substrate marker of CYP2B6 catalytic activity.