HSD11B111%CE%B2-Hydroxysteroid-Dehydrogenase_111%CE%B2-Hydroxysteroid_dehydrogenase_type_111%CE%B2-Hydroxyst%C3%A9ro%C3%AFde_d%C3%A9shydrog%C3%A9nase_1Dehydrogenaza_11%CE%B2-hydroksysteroidowa_typu_111%CE%B2-hidroxiesteroide_desidrogenase_tipo_111-%D0%B1%D0%B5%D1%82%D0%B0-%D0%B3%D0%B8%D0%B4%D1%80%D0%BE%D0%BA%D1%81%D0%B8%D1%81%D1%82%D0%B5%D1%80%D0%BE%D0%B8%D0%B4%D0%B4%D0%B5%D0%B3%D0%B8%D0%B4%D1%80%D0%BE%D0%B3%D0%B5%D0%BD%D0%B0%D0%B7%D0%B0_1-%D0%B3%D0%BE_%D1%82%D0%B8%D0%BF%D0%B0HSD11B1Q17160411%CE%B2-%E7%BE%9F%E5%9F%BA%E7%B1%BB%E5%9B%BA%E9%86%87%E8%84%B1%E6%B0%A2%E9%85%B61%E5%9E%8B
about
P1855
P527
P688
Appropriate function of 11beta-hydroxysteroid dehydrogenase type 1 in the endoplasmic reticulum lumen is dependent on its N-terminal region sharing similar topological determinants with 50-kDa esteraseThe discovery of 2-anilinothiazolones as 11beta-HSD1 inhibitorsStructural characterization and pharmacodynamic effects of an orally active 11beta-hydroxysteroid dehydrogenase type 1 inhibitorPyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo modelDiscovery and optimization of piperidyl benzamide derivatives as a novel class of 11beta-HSD1 inhibitorsThe N-terminal anchor sequences of 11beta-hydroxysteroid dehydrogenases determine their orientation in the endoplasmic reticulum membraneConformational flexibility in crystal structures of human 11beta-hydroxysteroid dehydrogenase type I provide insights into glucocorticoid interconversion and enzyme regulation.Adamantane sulfone and sulfonamide 11-beta-HSD1 Inhibitors.
P921
Q24293608-9D12F9A3-C894-4A2A-9CCE-458F0EBF8457Q27648722-9AA6CB7D-A274-4A99-9537-0FEAC07F39CDQ27649250-6E1F7F43-1081-4AE5-BEC7-18D61332AADFQ27650633-09921871-75A3-4CEE-919A-90E9792C9C13Q27650834-2C5FA2B2-6AAB-4657-AD0E-240850257FB5Q27653807-08B966AF-3E8F-482E-8BF8-6A01DB7D7174Q28144963-4C18F165-31F3-49B9-A69F-70C4061728C3Q45129829-AA3208CF-9370-4552-9265-3ADCBB8C007DQ48385767-745A7A0D-ABFD-476E-B64B-0A3073A8A312
P921
description
Protein
@de
mammalian protein found in Homo sapiens
@en
menselijk eiwit
@nl
protein
@id
protein
@sv
proteinë
@sq
protèin
@ace
protéine humaine
@fr
фермент человека
@ru
بروتين في الإنسان العاقل
@ar
name
11-бета-гидроксистероиддегидрогеназа 1-го типа
@ru
11beta-Hydroxysteroid-Dehydrogenase 1
@de
11β-hidroxiesteroide desidrogenase tipo 1
@pt
11β-hydroxysteroid dehydrogenase type 1
@fr
11β-羟基类固醇脱氢酶1型
@zh
Dehydrogenaza 11β-hydroksysteroidowa typu 1
@pl
HSD11B1
@cy
HSD11B1
@uk
Hydroxysteroid 11-beta dehydrogenase 1
@en
Hydroxysteroid 11-beta dehydrogenase 1
@nl
type
label
11-бета-гидроксистероиддегидрогеназа 1-го типа
@ru
11beta-Hydroxysteroid-Dehydrogenase 1
@de
11β-hidroxiesteroide desidrogenase tipo 1
@pt
11β-hydroxysteroid dehydrogenase type 1
@fr
11β-羟基类固醇脱氢酶1型
@zh
Dehydrogenaza 11β-hydroksysteroidowa typu 1
@pl
HSD11B1
@cy
HSD11B1
@uk
Hydroxysteroid 11-beta dehydrogenase 1
@en
Hydroxysteroid 11-beta dehydrogenase 1
@nl
altLabel
11-DH
@en
11-beta-HSD1
@en
11-beta-hydroxysteroid dehydrogenase 1
@en
HSD11B1
@en
corticosteroid 11-beta-dehydrogenase isozyme 1
@en
short chain dehydrogenase/reductase family 26C member 1
@en
prefLabel
11-бета-гидроксистероиддегидрогеназа 1-го типа
@ru
11beta-Hydroxysteroid-Dehydrogenase 1
@de
11β-hidroxiesteroide desidrogenase tipo 1
@pt
11β-hydroxysteroid dehydrogenase type 1
@fr
11β-羟基类固醇脱氢酶1型
@zh
Dehydrogenaza 11β-hydroksysteroidowa typu 1
@pl
HSD11B1
@cy
HSD11B1
@uk
Hydroxysteroid 11-beta dehydrogenase 1
@en
Hydroxysteroid 11-beta dehydrogenase 1
@nl
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P2888
P31
P352
P486
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NP_001193670
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ENSP00000261465
ENSP00000355994
ENSP00000355995
ENSP00000478430