The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist - sprookjes - yvandenbroek - TriplyDB

The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

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Differential modulation of Beta-adrenergic receptor signaling by trace amine-associated receptor 1 agonists Structure of an agonist-bound human A2A adenosine receptor Agonist-bound adenosine A2A receptor structures reveal common features of GPCR activation Structural basis for the binding of the membrane-proximal C-terminal region of chemokine receptor CCR2 with the cytosolic regulator FROUNT Crystal structure of a lipid G protein-coupled receptor Structure of the human κ-opioid receptor in complex with JDTic Identification of three residues essential for 5-hydroxytryptamine 2A-metabotropic glutamate 2 (5-HT2A·mGlu2) receptor heteromerization and its psychoactive behavioral function Structural model of ligand-G protein-coupled receptor (GPCR) complex based on experimental double mutant cycle data: MT7 snake toxin bound to dimeric hM1 muscarinic receptor Structure of the human histamine H1 receptor complex with doxepin Structure of a nanobody-stabilized active state of the β(2) adrenoceptor Structure of the human glucagon class B G-protein-coupled receptor Structures of the CXCR4 chemokine GPCR with small-molecule and cyclic peptide antagonists The impact of GPCR structures on pharmacology and structure-based drug design Structure of the human M2 muscarinic acetylcholine receptor bound to an antagonist GPRC6A mediates the non-genomic effects of steroids.G protein-coupled receptors in the hypothalamic paraventricular and supraoptic nuclei--serpentine gateways to neuroendocrine homeostasis Identification of two distinct inactive conformations of the beta2-adrenergic receptor reconciles structural and biochemical observations G Protein-Coupled Receptors (GPCRs) in Alzheimer's Disease: A Focus on BACE1 Related GPCRs Charting a Path to Success in Virtual Screening Structural Studies of G Protein-Coupled Receptors Post-expression strategies for structural investigations of membrane proteins.Diversity and modularity of G protein-coupled receptor structures Large-scale production and protein engineering of G protein-coupled receptors for structural studies To fuse or not to fuse: what is your purpose?New insights for drug design from the X-ray crystallographic structures of G-protein-coupled receptors Fluorescent approaches for understanding interactions of ligands with G protein coupled receptors Tools for GPCR drug discovery.Endogenous lipid activated G protein-coupled receptors: emerging structural features from crystallography and molecular dynamics simulations Turning receptors on and off with intracellular pepducins: new insights into G-protein-coupled receptor drug development Cardiac contractility structure-activity relationship and ligand-receptor interactions; the discovery of unique and novel molecular switches in myosuppressin signaling Communication over the network of binary switches regulates the activation of A2A adenosine receptor Molecular modeling of the human P2Y14 receptor: A template for structure-based design of selective agonist ligands.Membrane-sensitive conformational states of helix 8 in the metabotropic Glu2 receptor, a class C GPCR Induced effects of sodium ions on dopaminergic G-protein coupled receptors A new drug design targeting the adenosinergic system for Huntington's disease Ligand-specific regulation of the extracellular surface of a G-protein-coupled receptor Structure of a Double Transmembrane Fragment of a G-Protein-Coupled Receptor in Micelles Structure determination of the seven-helix transmembrane receptor sensory rhodopsin II by solution NMR spectroscopy Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist Two distinct conformations of helix 6 observed in antagonist-bound structures of a 1-adrenergic receptor

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The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

http://www.wikidata.org/entity/Q24654563

description

2008 nî lūn-bûn

@nan

2008 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած

@hyw

2008 թվականի նոյեմբերին հրատարակված գիտական հոդված

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2008年の論文

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2008年論文

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2008年論文

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2008年論文

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2008年論文

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2008年論文

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2008年论文

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The 2.6 angstrom crystal struc ...... eceptor bound to an antagonist

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The 2.6 angstrom crystal struc ...... eceptor bound to an antagonist

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SCIENCE.1164772

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The 2.6 angstrom crystal struc ...... eceptor bound to an antagonist

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Ellen Y T Chien

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J Robert Lane

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Mark T Griffith

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Michael A Hanson

http://www.w3.org/2001/XMLSchema#string

P2860

Site-directed mutagenesis identifies residues involved in ligand recognition in the human A2a adenosine receptor

Adenosine receptors as therapeutic targets

Adenosine receptors and asthma.

The A(2A)-adenosine receptor: a GPCR with unique features?

High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor

The G protein-coupled receptor repertoires of human and mouse

Crystal structure of rhodopsin: A G protein-coupled receptor

Thermodynamic and structural studies of cavity formation in proteins suggest that loss of packing interactions rather than the hydrophobic effect dominates the observed energetics

Crystal structure of the human beta2 adrenergic G-protein-coupled receptor

Crystal structure of squid rhodopsin

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1211-7

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scholarly article

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2590909

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10.1126/SCIENCE.1164772

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5905

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322

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Raymond C Stevens

Adriaan P IJzerman

Veli-Pekka Jaakola

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2008-11-21T00:00:00Z

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23297175

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18832607

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crystal structure

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2586971

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