The sigma-receptor antagonist BD-1063 decreases ethanol intake and reinforcement in animal models of excessive drinking
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Targeting sigma receptors: novel medication development for drug abuse and addictionReinforcing effects of sigma-receptor agonists in rats trained to self-administer cocaineDifferential changes in amygdala and frontal cortex Pde10a expression during acute and protracted withdrawalCRF mediates the anxiogenic and anti-rewarding, but not the anorectic effects of PACAPAnimal models for medications development targeting alcohol abuse using selectively bred rat lines: neurobiological and pharmacological validityOperant alcohol self-administration in dependent rats: focus on the vapor modelCorticotropin releasing factor-induced amygdala gamma-aminobutyric Acid release plays a key role in alcohol dependence.High trait impulsivity predicts food addiction-like behavior in the ratTargeting ligand-operated chaperone sigma-1 receptors in the treatment of neuropsychiatric disorders.Activation of σ-receptors induces binge-like drinking in Sardinian alcohol-preferring ratsSigma-1 receptor mediates acquisition of alcohol drinking and seeking behavior in alcohol-preferring rats.Antagonism of sigma-1 receptors blocks compulsive-like eating.Ethanol-related behaviors in mice lacking the sigma-1 receptorThe lifetime of UDP-galactose:ceramide galactosyltransferase is controlled by a distinct endoplasmic reticulum-associated degradation (ERAD) regulated by sigma-1 receptor chaperonesThe uncompetitive NMDA receptor antagonists ketamine and memantine preferentially increase the choice for a small, immediate reward in low-impulsive ratsThe sigma-1 receptor: roles in neuronal plasticity and diseasemTOR activation is required for the anti-alcohol effect of ketamine, but not memantine, in alcohol-preferring ratsOpioid system in the medial prefrontal cortex mediates binge-like eatingSigma-1 receptor knockout mice display a depressive-like phenotype.Selective reduction of alcohol drinking in Sardinian alcohol-preferring rats by a sigma-1 receptor antagonist.Withdrawal from chronic, intermittent access to a highly palatable food induces depressive-like behavior in compulsive eating rats.A modified adjusting delay task to assess impulsive choice between isocaloric reinforcers in non-deprived male rats: effects of 5-HT₂A/C and 5-HT₁A receptor agonists.Pathological Overeating: Emerging Evidence for a Compulsivity Construct.Rat animal models for screening medications to treat alcohol use disorders.Sigma Receptors and Substance Use Disorders.Dysregulation of Brain Stress Systems Mediates Compulsive Alcohol Drinking.Pituitary adenylate cyclase-activating polypeptide (PACAP) in the central nucleus of the amygdala induces anxiety via melanocortin receptors.The Sigma-2 Receptor Selective Agonist Siramesine (Lu 28-179) Decreases Cocaine-Reinforced Pavlovian Learning and Alters Glutamatergic and Dopaminergic Input to the Striatum.A behavioral and pharmacological characterization of palatable diet alternation in mice.Infusion of brain-derived neurotrophic factor into the ventral tegmental area switches the substrates mediating ethanol motivation.Sigma Receptors and Alcohol Use Disorders.
P2860
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P2860
The sigma-receptor antagonist BD-1063 decreases ethanol intake and reinforcement in animal models of excessive drinking
description
2009 nî lūn-bûn
@nan
2009 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
name
The sigma-receptor antagonist ...... l models of excessive drinking
@ast
The sigma-receptor antagonist ...... l models of excessive drinking
@en
The sigma-receptor antagonist ...... l models of excessive drinking
@nl
type
label
The sigma-receptor antagonist ...... l models of excessive drinking
@ast
The sigma-receptor antagonist ...... l models of excessive drinking
@en
The sigma-receptor antagonist ...... l models of excessive drinking
@nl
prefLabel
The sigma-receptor antagonist ...... l models of excessive drinking
@ast
The sigma-receptor antagonist ...... l models of excessive drinking
@en
The sigma-receptor antagonist ...... l models of excessive drinking
@nl
P2093
P2860
P50
P356
P1476
The sigma-receptor antagonist ...... l models of excessive drinking
@en
P2093
Eric P Zorrilla
George F Koob
Kenner C Rice
Malliga R Iyer
P2860
P2888
P304
P356
10.1038/NPP.2008.192
P407
P577
2009-05-01T00:00:00Z
P5875
P6179
1038272435