Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB1 among different membrane microenvironments.
about
Mapping Cannabinoid 1 Receptor Allosteric Site(s): Critical Molecular Determinant and Signaling Profile of GAT100, a Novel, Potent, and Irreversibly Binding Probe.Allosteric Modulation: An Alternate Approach Targeting the Cannabinoid CB1 Receptor.In silico mapping of allosteric ligand binding sites in type-1 cannabinoid receptor.Role of palmitoylation of cysteine 415 in functional coupling CB1 receptor to Gαi2 protein.Leveraging allostery to improve G protein-coupled receptor (GPCR)-directed therapeutics: cannabinoid receptor 1 as discovery target.Modulation of CB1 cannabinoid receptor by allosteric ligands: Pharmacology and therapeutic opportunities.Effect of N-arachidonoyl-l-serine on human cerebromicrovascular endothelium.Assessing Allosteric Modulation of CB1 at the Receptor and Cellular Levels.Allosteric modulators of cannabinoid receptor 1: developing compounds for improved specificity.Homology Modeling, Validation and Dynamics of the G Protein-coupled Estrogen Receptor 1 (GPER-1).
P2860
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P2860
Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB1 among different membrane microenvironments.
description
2015 nî lūn-bûn
@nan
2015 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2015 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
name
Endogenous vs Exogenous Allost ...... ent membrane microenvironments
@nl
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@ast
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@en
type
label
Endogenous vs Exogenous Allost ...... ent membrane microenvironments
@nl
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@ast
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@en
prefLabel
Endogenous vs Exogenous Allost ...... ent membrane microenvironments
@nl
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@ast
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@en
P2093
P2860
P50
P356
P1433
P1476
Endogenous vs Exogenous Allost ...... nt membrane microenvironments.
@en
P2093
Agostino Bruno
Lorenzo Botta
Luciana Marinelli
Romano Silvestri
P2860
P2888
P356
10.1038/SREP15453
P407
P577
2015-10-20T00:00:00Z
P5875
P6179
1019923809