Mechanistic and Structural Analysis of Aminoglycoside N -Acetyltransferase AAC(6′)-Ib and Its Bifunctional, Fluoroquinolone-Active AAC(6′)-Ib-cr Variant † ‡
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Plasmid-mediated quinolone resistance: a multifaceted threatStructure and Functional Diversity of GCN5-Related N-Acetyltransferases (GNAT)Bacterial GCN5-Related N-Acetyltransferases: From Resistance to RegulationStrategies to overcome the action of aminoglycoside-modifying enzymes for treating resistant bacterial infectionsIdentification and characterization of a novel aac(6')-Iag associated with the blaIMP-1-integron in a multidrug-resistant Pseudomonas aeruginosaComparing aminoglycoside binding sites in bacterial ribosomal RNA and aminoglycoside modifying enzymes.Structure of the bifunctional aminoglycoside-resistance enzyme AAC(6')-Ie-APH(2'')-Ia revealed by crystallographic and small-angle X-ray scattering analysis.Aminoglycoside modifying enzymes.Structural and biochemical analysis of the pentapeptide repeat protein EfsQnr, a potent DNA gyrase inhibitorPlasmid-mediated quinolone resistance.Inhibitors of the aminoglycoside 6'-N-acetyltransferase type Ib [AAC(6')-Ib] identified by in silico molecular docking.Structural and molecular basis for resistance to aminoglycoside antibiotics by the adenylyltransferase ANT(2″)-IaSusceptibility of vertilmicin to modifications by three types of recombinant aminoglycoside-modifying enzymes.Structural characterization of a Gcn5-related N-acetyltransferase from Staphylococcus aureus.Purification, crystallization and preliminary X-ray analysis of the aminoglycoside-6'-acetyltransferase AAC(6')-Im.Identification of an Inhibitor of the Aminoglycoside 6'-N-Acetyltransferase type Ib [AAC(6')-Ib] by Glide Molecular DockingIdentification and characterization of inhibitors of the aminoglycoside resistance acetyltransferase Eis from Mycobacterium tuberculosisMechanisms of drug resistance: quinolone resistance.Prevalence of qnr and aac(6')-Ib-cr Genes in Clinical Isolates of Klebsiella Pneumoniae from Imam Hussein Hospital in Tehran.Global fluoroquinolone resistance epidemiology and implictions for clinical use.Cosubstrate tolerance of the aminoglycoside resistance enzyme Eis from Mycobacterium tuberculosisUnexpected N-acetylation of capreomycin by mycobacterial Eis enzymes.Rise and dissemination of aminoglycoside resistance: the aac(6')-Ib paradigm.High incidence of plasmid-mediated quinolone resistance genes among ciprofloxacin-resistant clinical isolates of Enterobacteriaceae at a tertiary care hospital in Puducherry, India.Novel resistance functions uncovered using functional metagenomic investigations of resistance reservoirsTemporal appearance of plasmid-mediated quinolone resistance genesComparative Study of Eis-like Enzymes from Pathogenic and Nonpathogenic Bacteria.Understanding and overcoming aminoglycoside resistance caused by N-6'-acetyltransferase.Topoisomerase Inhibitors: Fluoroquinolone Mechanisms of Action and Resistance.Effects of altering aminoglycoside structures on bacterial resistance enzyme activities.Small-angle X-ray scattering analysis of the bifunctional antibiotic resistance enzyme aminoglycoside (6') acetyltransferase-ie/aminoglycoside (2'') phosphotransferase-ia reveals a rigid solution structure.Tobramycin Variants with Enhanced Ribosome-Targeting ActivityMultiple keys for a single lock: the unusual structural plasticity of the nucleotidyltransferase (4')/kanamycin complex.Aminoglycoside resistance profile and structural architecture of the aminoglycoside acetyltransferase AAC(6')-Im.Comprehensive review of chemical strategies for the preparation of new aminoglycosides and their biological activities.Polymorphism of antibiotic-inactivating enzyme driven by ecology expands the environmental resistome.A low-barrier hydrogen bond mediates antibiotic resistance in a noncanonical catalytic triad.Plasticity of aminoglycoside binding to antibiotic kinase APH(2")-Ia.Aminoglycoside resistance in clinical Escherichia coli and Klebsiella pneumoniae isolates from Western Norway.Identification of Novel Protein Lysine Acetyltransferases in Escherichia coli
P2860
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P2860
Mechanistic and Structural Analysis of Aminoglycoside N -Acetyltransferase AAC(6′)-Ib and Its Bifunctional, Fluoroquinolone-Active AAC(6′)-Ib-cr Variant † ‡
description
2008 nî lūn-bûn
@nan
2008 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@ast
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@en
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@nl
type
label
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@ast
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@en
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@nl
prefLabel
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@ast
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@en
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@nl
P2093
P2860
P3181
P356
P1433
P1476
Mechanistic and Structural Ana ...... tive AAC(6′)-Ib-cr Variant † ‡
@en
P2093
Chi Hye Park
David C Hooper
George A Jacoby
John S Blanchard
Matthew W Vetting
Subray S Hegde
P2860
P304
P3181
P356
10.1021/BI800664X
P407
P577
2008-09-16T00:00:00Z