Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
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Structure and Functional Diversity of GCN5-Related N-Acetyltransferases (GNAT)Strategies to overcome the action of aminoglycoside-modifying enzymes for treating resistant bacterial infectionsMycobacterium tuberculosis Eis protein initiates suppression of host immune responses by acetylation of DUSP16/MKP-7Chemical and Structural Insights into the Regioversatility of the Aminoglycoside Acetyltransferase EisPotent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosisOctanoylation of early intermediates of mycobacterial methylglucose lipopolysaccharidesA random sequential mechanism of aminoglycoside acetylation by Mycobacterium tuberculosis Eis proteinMolecular characterization of amikacin, kanamycin and capreomycin resistance in M/XDR-TB strains isolated in Thailand.New trends in aminoglycosides use.Thermostable hexameric form of Eis (Rv2416c) protein of M. tuberculosis plays an important role for enhanced intracellular survival within macrophagesStructure of Mycobacterium smegmatis Eis in complex with paromomycinDiscovery of a new ATP-binding motif involved in peptidic azoline biosynthesis.Rapid synthesis, RNA binding, and antibacterial screening of a peptidic-aminosugar (PA) libraryInfluence of linker length and composition on enzymatic activity and ribosomal binding of neomycin dimers.Inhibition of aminoglycoside acetyltransferase resistance enzymes by metal salts.Amphiphilic Tobramycin Analogues as Antibacterial and Antifungal Agents.Microevolution of extensively drug-resistant tuberculosis in Russia.Identification and characterization of inhibitors of the aminoglycoside resistance acetyltransferase Eis from Mycobacterium tuberculosisAminoglycoside multiacetylating activity of the enhanced intracellular survival protein from Mycobacterium smegmatis and its inhibition.Synthesis and Biological Activity of Mono- and Di-N-acylated Aminoglycosides.Biochemical and structural analysis of an Eis family aminoglycoside acetyltransferase from bacillus anthracis.Cosubstrate tolerance of the aminoglycoside resistance enzyme Eis from Mycobacterium tuberculosisBiochemical and structural analysis of aminoglycoside acetyltransferase Eis from Anabaena variabilisArginine-linked neomycin B dimers: synthesis, rRNA binding, and resistance enzyme activity.Mechanisms of Resistance to Aminoglycoside Antibiotics: Overview and PerspectivesUnexpected N-acetylation of capreomycin by mycobacterial Eis enzymes.A review of patents (2011-2015) towards combating resistance to and toxicity of aminoglycosidesRise and dissemination of aminoglycoside resistance: the aac(6')-Ib paradigm.Redesign of substrate specificity and identification of the aminoglycoside binding residues of Eis from Mycobacterium tuberculosis.Overexpression of the Rv0805 phosphodiesterase elicits a cAMP-independent transcriptional responseTranscriptional Profiling of Mycobacterium tuberculosis Exposed to In Vitro Lysosomal Stress.Synthesis and evaluation of hetero- and homodimers of ribosome-targeting antibiotics: antimicrobial activity, in vitro inhibition of translation, and drug resistance.Comparative Study of Eis-like Enzymes from Pathogenic and Nonpathogenic Bacteria.Synthesis and Bioactivities of Kanamycin B-Derived Cationic Amphiphiles.Understanding and overcoming aminoglycoside resistance caused by N-6'-acetyltransferase.WhiB7, a transcriptional activator that coordinates physiology with intrinsic drug resistance in Mycobacterium tuberculosis.Advances In Mycobacterium Tuberculosis Therapeutics Discovery Utlizing Structural Biology.Molecular biology of drug resistance in Mycobacterium tuberculosisResistance in tuberculosis: what do we know and where can we go?First Insight Into the Fluoroquinolone and Aminoglycoside Resistance of Multidrug-Resistant Mycobacterium tuberculosis in Saudi Arabia.
P2860
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P2860
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
description
2011 nî lūn-bûn
@nan
2011 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@ast
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@en
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@nl
type
label
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@ast
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@en
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@nl
prefLabel
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@ast
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@en
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@nl
P2093
P2860
P3181
P356
P1476
Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB
@en
P2093
Oleg V Tsodikov
Tapan Biswas
Vanessa R Porter
Wenjing Chen
P2860
P304
P3181
P356
10.1073/PNAS.1105379108
P407
P577
2011-06-14T00:00:00Z