Generation of Candidate Ligands for Nicotinic Acetylcholine Receptors via in situ Click Chemistry with a Soluble Acetylcholine Binding Protein Template
about
In situ click chemistry: from small molecule discovery to synthetic antibodiesAssembly of a π–π stack of ligands in the binding site of an acetylcholine-binding proteinObservation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitorKinetic target-guided synthesis in drug discovery and chemical biology: a comprehensive facts and figures surveyReal time ligand-induced motion mappings of AChBP and nAChR using X-ray single molecule trackingIn situ click chemistry generation of cyclooxygenase-2 inhibitors.A chemical epitope-targeting strategy for protein capture agents: the serine 474 epitope of the kinase Akt2.Cholate-based synthesis of size-tunable cage compoundsSynthesis of selective agonists for the α7 nicotinic acetylcholine receptor with in situ click-chemistry on acetylcholine-binding protein templates.New insights into the kinetic target-guided synthesis of protein ligands.Structural Studies of Nicotinic Acetylcholine Receptors: Using Acetylcholine-Binding Protein as a Structural Surrogate.Ribosome-Templated Azide-Alkyne Cycloadditions: Synthesis of Potent Macrolide Antibiotics by In Situ Click Chemistry.Probing the binding site of abl tyrosine kinase using in situ click chemistry.Selective RNA versus DNA G-quadruplex targeting by in situ click chemistry.Reaction site-driven regioselective synthesis of AChE inhibitors.Optimising in situ click chemistry: the screening and identification of biotin protein ligase inhibitors
P2860
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P2860
Generation of Candidate Ligands for Nicotinic Acetylcholine Receptors via in situ Click Chemistry with a Soluble Acetylcholine Binding Protein Template
description
2012 nî lūn-bûn
@nan
2012 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Generation of Candidate Ligand ...... oline Binding Protein Template
@ast
Generation of Candidate Ligand ...... oline Binding Protein Template
@en
Generation of Candidate Ligand ...... oline Binding Protein Template
@nl
type
label
Generation of Candidate Ligand ...... oline Binding Protein Template
@ast
Generation of Candidate Ligand ...... oline Binding Protein Template
@en
Generation of Candidate Ligand ...... oline Binding Protein Template
@nl
prefLabel
Generation of Candidate Ligand ...... oline Binding Protein Template
@ast
Generation of Candidate Ligand ...... oline Binding Protein Template
@en
Generation of Candidate Ligand ...... oline Binding Protein Template
@nl
P2093
P2860
P356
P1476
Generation of Candidate Ligand ...... oline Binding Protein Template
@en
P2093
Bernhard Stump
John G Yamauchi
Joseph R Fotsing
Kwok-Yiu Ho
Neil P Grimster
Palmer Taylor
Timo Weide
Todd T Talley
Ákos Nemecz
P2860
P304
P356
10.1021/JA3001858
P407
P577
2012-04-18T00:00:00Z