R -Configuration of 4-Aminopyridyl-Based Inhibitors of CYP51 Confers Superior Efficacy Against Trypanosoma cruzi
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Expanding the Binding Envelope of CYP51 Inhibitors TargetingTrypanosoma cruziwith 4-Aminopyridyl-Based Sulfonamide Derivatives4-Aminopyridyl-Based CYP51 Inhibitors as Anti- Trypanosoma cruzi Drug Leads with Improved Pharmacokinetic Profile and in Vivo PotencyThe Potential of Secondary Metabolites from Plants as Drugs or Leads against Protozoan Neglected Diseases-Part III: In-Silico Molecular Docking InvestigationsTargeting Ergosterol biosynthesis in Leishmania donovani: essentiality of sterol 14 alpha-demethylaseMachine Learning Models and Pathway Genome Data Base for Trypanosoma cruzi Drug DiscoveryDrug strategies targeting CYP51 in neglected tropical diseasesBinding mode and potency of N-indolyloxopyridinyl-4-aminopropanyl-based inhibitors targeting Trypanosoma cruzi CYP51.Fragment-Based Approaches to the Development of Mycobacterium tuberculosis CYP121 Inhibitors.4-aminopyridyl-based lead compounds targeting CYP51 prevent spontaneous parasite relapse in a chronic model and improve cardiac pathology in an acute model of Trypanosoma cruzi infection.
P2860
Q27683570-06D21709-63F8-4246-BC81-0C077109FEACQ27684956-840624E7-4DA1-4A39-AD10-07AF230AD3FCQ28066944-26B0817A-5E55-48FC-B1CF-33FA54A20BDDQ28544037-0FDAC276-26BE-404A-AE6E-7B6F7402AE37Q28545842-77C7366B-3BFF-44C6-BA46-1F0ABE88AADDQ34622554-253FCDA2-AEDD-49A1-944D-690B9606B67BQ34701325-D4EC68FF-C5B1-4FB3-B521-42156D44289AQ36808252-81E0AF9E-D02F-44D2-A0A4-93F7964B7355Q48342608-2E065E15-90A7-43DE-B9B2-694E12796BE8
P2860
R -Configuration of 4-Aminopyridyl-Based Inhibitors of CYP51 Confers Superior Efficacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
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P2093
P2860
P921
P3181
P356
P1476
R -Configuration of 4-Aminopyr ...... cacy Against Trypanosoma cruzi
@en
P2093
Claudia M Calvet
Debora F Vieira
Jun Yong Choi
Larissa M Podust
Michael D Cameron
Shamila S Gunatilleke
William R Roush
P2860
P3181
P356
10.1021/ML500010M
P577
2014-04-10T00:00:00Z