Structure of a glutamate-receptor ligand-binding core in complex with kainate
about
General anaesthetic actions on ligand-gated ion channelsKainate receptors coming of age: milestones of two decades of researchPiracetam defines a new binding site for allosteric modulators of alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA) receptorsCrystal structure of the ectodomain of Methuselah, a Drosophila G protein-coupled receptor associated with extended lifespanAmino acid substitutions in the pore helix of GluR6 control inhibition by membrane fatty acidsTargeting AMPA receptor gating processes with allosteric modulators and mutationsNovel NMDA receptor modulators: an updateSize matters in activation/inhibition of ligand-gated ion channelsMechanism of glutamate receptor desensitizationCrystal structure and mechanism of a calcium-gated potassium channelGluR2 ligand-binding core complexes: importance of the isoxazolol moiety and 5-substituent for the binding mode of AMPA-type agonistsTuning activation of the AMPA-sensitive GluR2 ion channel by genetic adjustment of agonist-induced conformational changesMechanisms of activation, inhibition and specificity: crystal structures of the NMDA receptor NR1 ligand-binding coreCrystal structure of a histidine kinase sensor domain with similarity to periplasmic binding proteinsMolecular mechanism of ligand recognition by NR3 subtype glutamate receptors6-Azido-7-nitro-1,4-dihydroquinoxaline-2,3-dione (ANQX) Forms an Irreversible Bond To the Active Site of the GluR2 AMPA Receptor †Structure of the S1S2 glutamate binding domain of GLuR3Mechanisms of Antagonism of the GluR2 AMPA Receptor: Structure and Dynamics of the Complex of Two Willardiine Antagonists with the Glutamate Binding DomainCrystal structure and association behaviour of the GluR2 amino-terminal domainThe N-terminal domain of GluR6-subtype glutamate receptor ion channelsX-ray structure, symmetry and mechanism of an AMPA-subtype glutamate receptorCrystal structure of the glutamate receptor GluA1 N-terminal domainStructural and Functional Analysis of Two New Positive Allosteric Modulators of GluA2 Desensitization and DeactivationMechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONSStructural Determinants of Agonist Efficacy at the Glutamate Binding Site of N-Methyl-D-Aspartate ReceptorsThe Loss of an Electrostatic Contact Unique to AMPA Receptor Ligand Binding Domain 2 Slows Channel ActivationMolecular actions of smoking cessation drugs at 4 2 nicotinic receptors defined in crystal structures of a homologous binding proteinStructure and functional interaction of the extracellular domain of human GABAB receptor GBR2Functional analysis of a novel positive allosteric modulator of AMPA receptors derived from a structure-based drug design strategyActivation of NMDA receptors and the mechanism of inhibition by ifenprodil.Modulation of non-NMDA receptor gating by auxiliary subunitsMolecular cloning and functional identification of mouse vesicular glutamate transporter 3 and its expression in subsets of novel excitatory neuronsAlpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor channels lacking the N-terminal domainGlutamate receptor ion channels: structure, regulation, and functionAncient protostome origin of chemosensory ionotropic glutamate receptors and the evolution of insect taste and olfactionInfluence of a threonine residue in the S2 ligand binding domain in determining agonist potency and deactivation rate of recombinant NR1a/NR2D NMDA receptorsMolecular determinants of coordinated proton and zinc inhibition of N-methyl-D-aspartate NR1/NR2A receptorsVariant ionotropic glutamate receptors as chemosensory receptors in DrosophilaSOL-1 is a CUB-domain protein required for GLR-1 glutamate receptor function in C. elegans.Overview of protein structural and functional folds.
P2860
Q24595524-2170DC5B-CDE5-42F8-87B4-8C0EABD79DF7Q24606030-035073CB-71B4-49A7-8A46-F63243A73495Q24611731-58614782-184C-43B8-A67F-2D8934CFB869Q24616895-537FFD43-3AFC-4CE1-AB13-78017A8A9011Q24648841-268247E2-E8EB-46AC-9C7D-D5C53BE66324Q24673639-73B57B8D-4B7A-4E73-B607-95541DE14C3CQ26849614-C619C298-D72D-4896-84EC-CD871CDDE36AQ27008299-B313EF7B-ADF6-4801-8A70-830441954388Q27639007-2068118F-55CA-462E-836E-6B35F5F6E8DBQ27639064-6744BCA8-BA28-49B3-8714-C4A52A9F0E34Q27639914-10994EDA-F061-47E1-BAB9-E8CA02862F4CQ27641132-EC0C4A53-FE84-476E-94AF-8F4A05A781ABQ27641433-5FBCE6C1-60E0-40E6-A2D3-D388B76140BAQ27643947-BEE7C783-075F-4E2F-8955-8EBE53494050Q27651229-FE7A783C-5522-4271-9B6E-BE9C490E5483Q27651830-D998C423-CEA2-4282-A339-31097FDF90A2Q27652871-03D2D320-2CDF-4B9C-8BB0-5B2B4F54168FQ27654089-E32834ED-10DC-442F-9A7C-2752B5BFA76CQ27655567-7ACDD5E2-9C6D-4E44-86EF-6C4DB9346A40Q27655599-EFC48C54-C2D6-4CC8-B42D-B3AB75117D68Q27658372-E717BDFD-EF68-4D32-AF70-EC15BAF13195Q27666247-246E35DB-74B9-45AE-BB61-85A515567A3DQ27667701-0538B635-DFE0-477B-A020-E23A5B65BE32Q27671791-2C84C2D2-ABB6-47F6-AB72-7BCC98358448Q27677835-F5650062-512C-4A42-9766-1E954C78305EQ27678596-4B5865D0-C22F-4EDA-ADD2-012F42FDB54FQ27679259-C6958E7B-BB15-48D8-B6FC-E9C842F7AE42Q27679465-50E72BC8-19C2-4DED-BAE0-7B5CB6A61EE9Q27681406-2A569954-A82A-478A-B6D6-AD1996E6D20BQ27704785-A86F2CC0-CB62-43C8-BC86-EA27F5D0C958Q28085008-044B4AF3-9D49-45E7-9499-5BE564F28EB9Q28207970-3F024B64-8EC5-481A-AB32-F364BC4F603DQ28210064-2465D285-FDB2-4CFA-9E2B-E319752DF307Q28290774-8314C9CE-C4F4-4914-AC7D-178CAD4D9636Q28475205-3A17C4A5-97D9-410D-AD78-DA6F5418307EQ28576339-CB89819E-5DCF-4222-99FE-87A6F0E7F7ECQ28776368-F380C8B8-8B6D-4179-A8C4-23F7046F66DFQ29616617-49C6D331-FEE5-4201-B1B2-8155FA4BAF43Q30164297-37C958F1-2F95-4139-A78E-FA5B8BECF005Q30368988-96880C68-139B-4F61-966C-51CADE2F34DB
P2860
Structure of a glutamate-receptor ligand-binding core in complex with kainate
description
1998 nî lūn-bûn
@nan
1998 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1998 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
1998年の論文
@ja
1998年学术文章
@wuu
1998年学术文章
@zh-cn
1998年学术文章
@zh-hans
1998年学术文章
@zh-my
1998年学术文章
@zh-sg
1998年學術文章
@yue
name
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@ast
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@en
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@nl
type
label
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@ast
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@en
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@nl
prefLabel
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@ast
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@en
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@nl
P2093
P3181
P356
P1433
P1476
Structure of a glutamate-receptor ligand-binding core in complex with kainate
@en
P2093
P2888
P3181
P356
10.1038/27692
P407
P577
1998-10-29T00:00:00Z
P5875
P6179
1038931719