The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
about
New invMED1 element cis-activates human multidrug-related MDR1 and MVP genes, involving the LRP130 proteinIdentification of an endogenous ligand that activates pregnane X receptor-mediated sterol clearanceHow to calculate the dose of chemotherapyReduced fat mass in mice lacking orphan nuclear receptor estrogen-related receptor alphaBiology of PXR: role in drug-hormone interactionsRole of pregnane X receptor in chemotherapeutic treatmentNuclear receptors in bone physiology and diseasesTargeting xenobiotic receptors PXR and CAR in human diseasesRole of Nuclear Receptors in Central Nervous System Development and Associated DiseasesCrystal structure of the PXR–T1317 complex provides a scaffold to examine the potential for receptor antagonismJapanese-US common-arm analysis of paclitaxel plus carboplatin in advanced non-small-cell lung cancer: a model for assessing population-related pharmacogenomics.PXR variants: the impact on drug metabolism and therapeutic responsesCockayne syndrome group B protein (CSB) plays a general role in chromatin maintenance and remodelingHistone deacetylase inhibitors regulate P-gp expression in colorectal cancer via transcriptional activation and mRNA stabilizationUp-regulating CYP3A4 expression in C3A cells by transfection with a novel chimeric regulator of hPXR-p53-ADPregnane X receptor knockout mice display aging-dependent wearing of articular cartilageAlterations of chemotherapeutic pharmacokinetic profiles by drug-drug interactionsPregnane X receptor and natural products: beyond drug-drug interactionsTargeting multidrug resistance in cancerDifferent modalities of intercellular membrane exchanges mediate cell-to-cell p-glycoprotein transfers in MCF-7 breast cancer cells.Intestinal and hepatic expression of cytochrome P450s and mdr1a in rats with indomethacin-induced small intestinal ulcersFunctional evolution of the vitamin D and pregnane X receptors.Human pregnane X receptor is expressed in breast carcinomas, potential heterodimers formation between hPXR and RXR-alphaVon Hippel-Lindau-coupled and transcription-coupled nucleotide excision repair-dependent degradation of RNA polymerase II in response to trabectedin.Polymorphisms in SLCO1B3 and NR1I2 as genetic determinants of hematotoxicity of carboplatin and paclitaxel combination.The transcriptional regulation of the human CYP2C genesThe phytoestrogen coumestrol is a naturally occurring antagonist of the human pregnane X receptorXenobiotic, bile acid, and cholesterol transporters: function and regulation.Hybrid scoring and classification approaches to predict human pregnane X receptor activatorsSpecific antioxidant compounds differentially modulate cytotoxic activity of doxorubicin and cisplatin: in vitro and in vivo study.Sulfotransferase genes: regulation by nuclear receptors in response to xeno/endo-biotics.Activation of xenobiotic receptors: driving into the nucleus.Elucidating the 'Jekyll and Hyde' nature of PXR: the case for discovering antagonists or allosteric antagonists.Evolution of acquired resistance to anti-cancer therapy.The importance of discerning shape in molecular pharmacology.Nuclear receptors constitutive androstane receptor and pregnane X receptor ameliorate cholestatic liver injury.Reversing multidrug resistance by RNA interference through the suppression of MDR1 gene in human hepatoma cells.Ontogeny of human hepatic and intestinal transporter gene expression during childhood: age matters.Drug resistance in brain diseases and the role of drug efflux transporters.Expression, localization and polymorphisms of the nuclear receptor PXR in Barrett's esophagus and esophageal adenocarcinoma
P2860
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P2860
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
description
2001 nî lūn-bûn
@nan
2001 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2001 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2001年の論文
@ja
2001年論文
@yue
2001年論文
@zh-hant
2001年論文
@zh-hk
2001年論文
@zh-mo
2001年論文
@zh-tw
2001年论文
@wuu
name
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@ast
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@en
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@nl
type
label
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@ast
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@en
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@nl
prefLabel
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@ast
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@en
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@nl
P2093
P3181
P356
P1433
P1476
The orphan nuclear receptor SXR coordinately regulates drug metabolism and efflux
@en
P2093
B M Forman
I Dussault
T W Synold
P2888
P304
P3181
P356
10.1038/87912
P407
P577
2001-05-01T00:00:00Z
P5875
P6179
1004128811